SCHEMBL8108320

SCHEMBL8108320

O=C(O)Cc1ccccc1CCCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.57
HDAC8 Q9BY41 3/20 0.57
HDAC3 O15379 2/20 0.57
HDAC4 P56524 2/20 0.57
HDAC7 Q8WUI4 2/20 0.57
HDAC2 Q92769 2/20 0.57
HDAC10 Q969S8 2/20 0.57
HDAC11 Q96DB2 2/20 0.57
HDAC6 Q9UBN7 2/20 0.57
HDAC9 Q9UKV0 2/20 0.57
HDAC5 Q9UQL6 2/20 0.57
MAPK1 P28482 1/20 0.57
ADRA1A P35348 1/20 0.57
SLC6A3 Q01959 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
AKR1B1 P15121 2/20 0.54
MAPT P10636 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
BID P55957 1/20 0.50
BCL2L1 Q07817 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5076822 0.88 AKR1B1 (0.58) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL24661354 0.88 AKR1B1 (0.58) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL16312704 0.85 ALDH1A1 (0.53) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL29588181 0.83 HTR2A (0.58) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL28963713 0.83 HTR2A (0.58) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL11544667 0.82 AKR1B1 (0.55) ADRA1AAKR1B1MAPTHPGDTDP1
SCHEMBL7821192 0.82 AKR1B1 (0.74) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL29410826 0.81 AKR1B1 (0.76) ADRA1AAKR1B1MAPTHPGDGAA
SCHEMBL30359 0.81 AKR1B1 (0.76) ADRA1AAKR1B1MAPTHPGDGAA
SCHEMBL10533147 0.81 AKR1B1 (0.53) ADRA1AAKR1B1MAPTRXFP1BID

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136819-A COMPOUNDS FOR ANTIINFLAMMATORY AGENTS OR CARDIOVASCULAR DISORDERS BOEHRINGER INGELHEIM GMBH (DE) 2000-10-24 US disclosed
EP-0736011-B1 ANELLATED DIHYDROPYRIDINES AND THEIR USE IN THE PRODUCTION OF PHARMACEUTICAL PREPARATIONS BOEHRINGER INGELHEIM INT (DE) 2000-07-26 EP disclosed
US-5968948-A FOR TREATMENT OF EPILEPSY, STROKE, ALZHEIMER'S DISEASE, BRAIN DISEASES OR AS ANTIINFLAMMATORY OR ANTIPROLIFERATIVE AGENTS BOERHINGER INGELHEIM GMBH (DE) 1999-10-19 US disclosed
US-5661157-A Annelated dihydropyridines and the use thereof for preparing pharmaceutical preparations BOEHRINGER INGELHEIM KG (DE) 1997-08-26 US disclosed
WO-1995017389-A1 ANELLATED DIHYDROPYRIDINES AND THEIR USE IN THE PRODUCTION OF PHARMACEUTICAL PREPARATIONS BOEHRINGER INGELHEIM KG (DE) 1995-06-29 WO disclosed