SCHEMBL8108416

SCHEMBL8108416

C[C@@H]1CN(c2ccc(F)c(Cl)c2)CCN1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2A1 Q16548 2/20 0.52
HSD11B1 P28845 1/20 0.48
MAPT P10636 2/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
KHK P50053 2/20 0.45
ADRB1 P08588 1/20 0.44
ACACB O00763 2/20 0.40
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
RAD51 Q06609 1/20 0.38
MMP2 P08253 1/20 0.38
ADAMTS5 Q9UNA0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8108460 0.88 BCL2A1 (0.55) BCL2A1HSD11B1MAPTALDH1A1LMNA
SCHEMBL18013225 0.86 BCL2A1 (0.66) BCL2A1HSD11B1MAPTALDH1A1LMNA
SCHEMBL8110875 0.86 MAPT (0.49) BCL2A1HSD11B1MAPTALDH1A1LMNA
SCHEMBL4936462 0.86 BCL2A1 (0.66) BCL2A1HSD11B1MAPTALDH1A1LMNA
SCHEMBL20159005 0.86 MAPT (0.49) BCL2A1HSD11B1MAPTALDH1A1LMNA
SCHEMBL8108419 0.85 BCL2A1 (0.54) BCL2A1HSD11B1MAPTALDH1A1LMNA
SCHEMBL8106618 0.84 KHK (0.49) BCL2A1HSD11B1MAPTALDH1A1LMNA
SCHEMBL1203360 0.81 HTR3E (0.56) BCL2A1MAPTALDH1A1LMNAKHK
SCHEMBL1203357 0.81 HTR3E (0.56) BCL2A1MAPTALDH1A1LMNAKHK
SCHEMBL2874784 0.81 HTR3E (0.56) BCL2A1MAPTALDH1A1LMNAKHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed