SCHEMBL8108842

SCHEMBL8108842

O=C1CCN(Cc2ccncc2)CC1.O=C1CCN(Cc2ccncc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.50
LSS P48449 1/20 0.50
KDM4E B2RXH2 4/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C9 P11712 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
HIF1A Q16665 1/20 0.49
POLB P06746 1/20 0.48
TNKS O95271 1/20 0.47
PARP1 P09874 1/20 0.47
PARP10 Q53GL7 1/20 0.47
TNKS2 Q9H2K2 1/20 0.47
PARP2 Q9UGN5 1/20 0.47
PARP4 Q9UKK3 1/20 0.47
PARP3 Q9Y6F1 1/20 0.47
DRD2 P14416 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4884441 1.00 HPGD (0.50) HPGDLSSKDM4ECYP3A4CYP2D6
SCHEMBL28269086 0.83 LSS (0.66) HPGDLSSKDM4ECYP3A4CYP2D6
SCHEMBL8356766 0.81 HRH3 (0.68) CYP3A4MEN1KMT2APOLBHRH3
SCHEMBL4726 0.80 SIGMAR1 (0.68) MEN1KMT2APOLBSIGMAR1
SCHEMBL3994683 0.79 HRH3 (0.67) HPGDLSSKDM4ECYP3A4CYP2D6
SCHEMBL8099601 0.79 CHRNB2 (0.70) KDM4EDRD2ALDH1A1OPRL1CASP1
SCHEMBL1830945 0.79 CHRNB2 (0.70) KDM4EDRD2ALDH1A1OPRL1CASP1
SCHEMBL941871 0.78 KDM4E (0.62) LSSKDM4EMEN1KMT2AHRH3
Hydrochloric Acid SCHEMBL5671727 0.78 SIGMAR1 (0.65) MEN1KMT2APOLBSIGMAR1
Iodide SCHEMBL1697595 0.78 SIGMAR1 (0.65) MEN1KMT2APOLBSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056744-A1 6,9-DISUBSTITUTED 2- TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES Aventis Pharmaceuticals Inc. (US) 2000-12-06 EP disclosed
WO-1999043675-A1 6,9-DISUBSTITUTED 2-[TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES AVENTIS PHARMACEUTICALS INC. (US) 1999-09-02 WO disclosed