SCHEMBL8109237

SCHEMBL8109237

NC1CCN(Cc2ccc(C(F)(F)F)cc2)CC1.NC1CCN(Cc2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.65
ALDH1A1 P00352 1/20 0.65
BCHE P06276 3/20 0.58
ACHE P22303 3/20 0.58
BACE1 P56817 3/20 0.58
TEAD1 P28347 2/20 0.54
SIGMAR1 Q99720 3/20 0.53
HIF1A Q16665 1/20 0.52
EPAS1 Q99814 1/20 0.52
CYP3A4 P08684 1/20 0.52
CHKA P35790 1/20 0.51
KCNH2 Q12809 1/20 0.51
MAOB P27338 1/20 0.50
DRD2 P14416 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
HTR2B P41595 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6941820 1.00 KDM4E (0.65) KDM4EALDH1A1BCHEACHEBACE1
SCHEMBL28600653 0.90 KDM4E (0.57) KDM4EALDH1A1BCHEACHEBACE1
SCHEMBL2734780 0.90 KDM4E (0.57) KDM4EALDH1A1BCHEACHEBACE1
SCHEMBL15223361 0.84 KDM4E (0.61) KDM4EALDH1A1BCHEACHEBACE1
Isophthalic Acid SCHEMBL27788675 0.83 SIGMAR1 (0.55) BCHEACHEBACE1TEAD1SIGMAR1
SCHEMBL14242820 0.83 HRH3 (0.67) KDM4EALDH1A1BCHEACHEBACE1
SCHEMBL6945302 0.83 CYP2D6 (0.52) KDM4EALDH1A1SIGMAR1HIF1ACYP3A4
SCHEMBL9139565 0.83 TEAD1 (0.53) KDM4EALDH1A1ACHETEAD1SIGMAR1
SCHEMBL1035980 0.83 ALDH1A1 (0.65) KDM4EALDH1A1BCHEACHEBACE1
Ammonia Solution, Strong SCHEMBL28813879 0.82 HRH3 (0.65) KDM4EALDH1A1BCHEACHEBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056744-A1 6,9-DISUBSTITUTED 2- TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES Aventis Pharmaceuticals Inc. (US) 2000-12-06 EP disclosed
WO-1999043675-A1 6,9-DISUBSTITUTED 2-[TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES AVENTIS PHARMACEUTICALS INC. (US) 1999-09-02 WO disclosed