SCHEMBL8109561

SCHEMBL8109561

CC1CN(c2ccccc2)C(=O)N(c2cccc(C(F)(F)F)c2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MAPK1 P28482 1/20 0.48
HSD17B10 Q99714 1/20 0.48
GRM2 Q14416 1/20 0.47
CYP17A1 P05093 1/20 0.46
DRD2 P14416 2/20 0.46
DRD3 P35462 2/20 0.46
KCNH2 Q12809 1/20 0.46
NOTUM Q6P988 1/20 0.46
OPRM1 P35372 1/20 0.46
OPRL1 P41146 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
RAB9A P51151 1/20 0.46
NFKB2 Q00653 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10987471 0.84 TSHR (0.51) ALDH1A1KDM4EHSD17B10CYP17A1SMN1; SMN2
SCHEMBL10965901 0.81 DRD2 (0.57) ALDH1A1CYP17A1DRD2DRD3KCNH2
SCHEMBL10983305 0.80 DRD2 (0.49) GRM2DRD2DRD3KCNH2NPC1
SCHEMBL10967325 0.79 ALDH1A1 (0.50) ALDH1A1KDM4EMAPK1HSD17B10CYP17A1
SCHEMBL10666765 0.78 MEN1 (0.46) ALDH1A1KDM4EMAPK1HSD17B10GRM2
SCHEMBL10988754 0.77 GRM2 (0.52) ALDH1A1GRM2DRD2DRD3TP53
SCHEMBL10988555 0.76 KMT2A (0.46) ALDH1A1MAPK1HSD17B10SMN1; SMN2NPC1
SCHEMBL10666890 0.75 DRD2 (0.46) ALDH1A1GRM2CYP17A1DRD2DRD3
SCHEMBL10988185 0.73 DRD2 (0.47) ALDH1A1KDM4EMAPK1HSD17B10DRD2
SCHEMBL11281751 0.72 DRD2 (0.52) ALDH1A1KDM4EMAPK1HSD17B10CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4514210-A Herbicidally active methyl-substituted tetrahydro-2-pyrimidinone derivatives NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1985-04-30 US claimed
EP-0585970-B1 Triazolin(thi)one intermediates for the preparation of herbicides BAYER AG (DE) 2000-10-18 EP disclosed
US-5750718-A CHEMICAL INTERMEDIATES BAYER AKTIENGESELLSCHAFT (DE) 1998-05-12 US disclosed
EP-0790242-A1 Substituted triazolinones BAYER AG (DE) 1997-08-20 EP disclosed
US-5599944-A Intermediates for herbicidal sulphonylaminocarbonyltriazolinones having substituents which are bonded via sulphur BAYER AKTIENGESELLSCHAFT (DE) 1997-02-04 US disclosed
US-5523409-A PREEMERGENCE, POSTEMERGENCE BAYER AKTIENGESELLSCHAFT (DE) 1996-06-04 US disclosed
EP-0283876-B1 Substituted triazolinones BAYER AG (DE) 1994-07-20 EP disclosed
EP-0585970-A2 Substituted triazolinones BAYER AG (DE) 1994-03-09 EP disclosed
US-5262389-A Substituted triazolinone herbicides and plant growth regulators BAYER AKTIENGESELLSCHAFT (DE) 1993-11-16 US disclosed
US-5166356-A Substituted triazolinone herbicides and plant growth regulators BAYER AKTIENGESELLSCHAFT (DE) 1992-11-24 US disclosed
US-5061311-A SUBSTITUTED TRIAZOLINONE HERBICIDES AND PLANT GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1991-10-29 US disclosed
EP-0283876-A2 Substituted triazolinones BAYER AG (DE) 1988-09-28 EP disclosed
US-4514210-A Herbicidally active methyl-substituted tetrahydro-2-pyrimidinone derivatives NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1985-04-30 US disclosed
EP-0137358-A2 1,3-Diaryl-5-methylene-perhydropyrimidin-2-one BAYER AG (DE) 1985-04-17 EP disclosed