SCHEMBL8110574

SCHEMBL8110574

CCCN1c2ccc(Cl)cc2C(c2ccccc2Cl)SCC1CC(=O)OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
TSHR P16473 2/20 0.37
CASP1 P29466 2/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
ALOX15 P16050 1/20 0.37
CYP2C19 P33261 1/20 0.37
RECQL P46063 1/20 0.37
SLC8B1 Q6J4K2 1/20 0.37
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
GLA P06280 2/20 0.36
GAA P10253 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
FFAR1 O14842 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8110758 0.85 MAPT (0.37) MAPTTSHRCASP1TP53CYP1A2
SCHEMBL8116269 0.74 MAPT (0.50) MAPTTSHRCASP1TP53CYP1A2
SCHEMBL8111295 0.73 ALDH1A1 (0.43) MAPTTSHRCYP2C9CYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL8110744 0.68 FDFT1 (0.41) MAPTTSHRCASP1TP53CYP1A2
SCHEMBL8103029 0.65 FDFT1 (0.39) MAPTTSHRCASP1TP53CYP1A2
SCHEMBL8112525 0.64 FDFT1 (0.42) MAPTTSHRCASP1TP53CYP1A2
SCHEMBL8110749 0.64 FDFT1 (0.44)
SCHEMBL8111693 0.63 FDFT1 (0.41) MAPTTSHRCASP1TP53CYP1A2
SCHEMBL38651042 0.62 NR1I2 (0.48) MAPTMEN1KMT2APTGDRPTGDR2
SCHEMBL8112208 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0645378-B1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-08-23 EP disclosed
US-5698691-A ANTICHOLESTEROL AGENT; SYNTHETASE INHIBITOR; FUNGICIDE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-12-16 US disclosed
EP-0645378-A1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors Takeda Chemical Industries, Ltd. (JP) 1995-03-29 EP disclosed