SCHEMBL8110758

SCHEMBL8110758

CCC(=O)N1c2ccc(Cl)cc2C(c2ccccc2Cl)SCC1CC(=O)OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
TSHR P16473 2/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
ALOX15 P16050 1/20 0.37
CASP1 P29466 1/20 0.37
CYP2C19 P33261 1/20 0.37
RECQL P46063 1/20 0.37
SLC8B1 Q6J4K2 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
PTGDR Q13258 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
ALDH1A1 P00352 1/20 0.35
PKM P14618 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.33
AVPR1A P37288 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8110574 0.85 MAPT (0.37) MAPTTSHRTP53CYP1A2CYP2C9
SCHEMBL8116269 0.74 MAPT (0.50) MAPTTSHRTP53CYP1A2CYP2C9
SCHEMBL8103029 0.70 FDFT1 (0.39) MAPTTSHRTP53CYP1A2CYP2C9
SCHEMBL8110749 0.64 FDFT1 (0.44) FDFT1
SCHEMBL8111804 0.63 FDFT1 (0.39) ADORA3FDFT1
SCHEMBL8111693 0.63 FDFT1 (0.41) MAPTTSHRTP53CYP1A2CYP2C9
Hydrochloric Acid SCHEMBL8110744 0.62 FDFT1 (0.41) MAPTTSHRTP53CYP1A2CYP2C9
SCHEMBL8112525 0.62 FDFT1 (0.42) MAPTTSHRTP53CYP1A2CYP2C9
SCHEMBL8111295 0.61 ALDH1A1 (0.43) MAPTTSHRCYP2C9CYP2C19SMN1; SMN2
SCHEMBL8110599 0.60 FDFT1 (0.43) MAPTTSHRTP53CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0645378-B1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-08-23 EP disclosed
US-5698691-A ANTICHOLESTEROL AGENT; SYNTHETASE INHIBITOR; FUNGICIDE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-12-16 US disclosed
EP-0645378-A1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors Takeda Chemical Industries, Ltd. (JP) 1995-03-29 EP disclosed