SCHEMBL8110643

SCHEMBL8110643

COc1c(I)cc(C(F)(F)F)cc1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.45
HSD17B10 Q99714 3/20 0.42
SORT1 Q99523 6/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
RXRA P19793 2/20 0.41
RXRB P28702 2/20 0.41
CYP2C19 P33261 2/20 0.41
USP2 O75604 1/20 0.41
AKR1C3 P42330 2/20 0.39
AKR1C2 P52895 2/20 0.39
ACLY P53396 1/20 0.38
CFTR P13569 1/20 0.37
NOTUM Q6P988 1/20 0.36
TAS2R14 Q9NYV8 1/20 0.36
RXRG P48443 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8118435 0.82 KDM4E (0.49) TPMTHSD17B10SORT1KDM4EALDH1A1
SCHEMBL22114934 0.82 HSD17B10 (0.44) HSD17B10SORT1KDM4EALDH1A1HPGD
SCHEMBL8116962 0.80 SLC9A1 (0.41) CFTR
Hydrochloric Acid SCHEMBL8110878 0.79 SLC9A1 (0.40) CFTR
SCHEMBL21609871 0.78 RXRA (0.47) HSD17B10SORT1KDM4EALDH1A1HPGD
SCHEMBL8116958 0.78 CFTR (0.36) TPMTSORT1KDM4ECYP2C19ACLY
SCHEMBL10370336 0.78 TPMT (0.51) TPMTHSD17B10KDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL8110876 0.77 CFTR (0.36) TPMTSORT1KDM4ECYP2C19ACLY
SCHEMBL24837048 0.76 TPMT (0.50) TPMTHSD17B10KDM4EALDH1A1HPGD
SCHEMBL16676482 0.75 KDM4E (0.50) HSD17B10KDM4EALDH1A1HPGDRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153651-A Ortho-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them HOECHST AKTIENGESELLSCHAFT (DE) 2000-11-28 US disclosed
EP-0794171-A2 Orthosubstituted benzoylguanidines, process for their preparation, their use as medicament or diagnostic material and medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1997-09-10 EP disclosed