SCHEMBL8111199

SCHEMBL8111199

C[C@@H](N1CCN(c2ccc(OCC(F)(F)C(F)F)cc2)C1=O)[C@@](O)(COS(C)(=O)=O)c1ccccc1F

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.34
LIPE Q05469 13/20 0.34
MMP13 P45452 1/20 0.33
MMP14 P50281 1/20 0.33
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
NOX4 Q9NPH5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8111197 1.00 ACACB (0.34) ACACBLIPEMMP13MMP14ALDH1A1
SCHEMBL8105653 0.89 ACACB (0.36) ACACBLIPEMMP13MMP14ALDH1A1
SCHEMBL8105650 0.89 ACACB (0.36) ACACBLIPEMMP13MMP14ALDH1A1
SCHEMBL6832831 0.83 CYP3A4 (0.39) ACACBLIPEHTT
SCHEMBL8106895 0.82 ACACB (0.32) ACACBMMP13MMP14ALDH1A1HTT
SCHEMBL8106891 0.82 ACACB (0.32) ACACBMMP13MMP14ALDH1A1HTT
SCHEMBL8540080 0.74 SCN9A (0.36) ACACBLIPEHTT
SCHEMBL8106760 0.74 CYP3A4 (0.49)
SCHEMBL8111015 0.73 PPARD (0.33)
SCHEMBL8111012 0.73 PPARD (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1033367-A2 Process for the preparation of optically active triazole derivatives and their imidazolidin-2-one intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-09-06 EP disclosed
US-5677464-A Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0687672-A2 Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-20 EP disclosed