SCHEMBL8112903

SCHEMBL8112903

CCOc1nc2cccc(C(=O)OCOC(=O)C(C)(C)C)c2n1Cc1ccc(-c2ccccc2-c2nnnn2C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 4/20 0.52
AGTR1 P30556 3/20 0.52
CYP3A4 P08684 2/20 0.52
ADORA3 P0DMS8 2/20 0.52
ADRA2B P18089 2/20 0.52
SLC6A2 P23975 2/20 0.52
PPARG P37231 2/20 0.52
HTR2B P41595 2/20 0.52
PDE3A Q14432 2/20 0.52
ABCB11 O95342 1/20 0.52
EGFR P00533 1/20 0.52
ERBB2 P04626 1/20 0.52
CYP2C9 P11712 1/20 0.52
ADRB3 P13945 1/20 0.52
TBXAS1 P24557 1/20 0.52
HTR2C P28335 1/20 0.52
LTB4R2 Q9NPC1 1/20 0.52
AGT P01019 1/20 0.45
NAE1 Q13564 4/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3873571 0.94 AGTR2 (0.56) AGTR2AGTR1CYP3A4ADORA3ADRA2B
SCHEMBL498030 0.89 AGTR1 (0.64) AGTR2AGTR1CYP3A4ADORA3ADRA2B
SCHEMBL9596667 0.88 AGTR1 (0.41) AGTR2AGTR1CYP3A4ADORA3ADRA2B
SCHEMBL28915096 0.88 AGTR2 (0.54) AGTR2AGTR1CYP3A4ADORA3ADRA2B
SCHEMBL8560666 0.84 AGTR2 (0.54) AGTR2AGTR1CYP3A4ADORA3ADRA2B
SCHEMBL10108979 0.84 AGTR1 (0.66) AGTR2AGTR1CYP3A4ADORA3ADRA2B
SCHEMBL7008517 0.84 AGTR1 (0.49) AGTR2AGTR1PPARGAGT
SCHEMBL1653579 0.84 AGTR2 (0.57) AGTR2AGTR1CYP3A4ADORA3ADRA2B
SCHEMBL166867 0.83 AGTR2 (0.56) AGTR2AGTR1CYP3A4ADORA3ADRA2B
SCHEMBL3429149 0.83 AGTR1 (0.57) AGTR2AGTR1CYP3A4ADORA3ADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668272-B1 A process for the production of tetrazolyl compounds TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-07-12 EP disclosed
US-5763619-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS OR STROKES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-09 US disclosed
US-5578733-A REACTION WITH MINERAL ACID IN THE PRESENCE OF ALCOHOL TO REMOVE PROTECTIVE GROUP TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-11-26 US disclosed
EP-0668272-A2 A process for the production of tetrazolyl compounds TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-23 EP disclosed