SCHEMBL8115331

SCHEMBL8115331

COc1cc(OC)c(OC)cc1C=Cc1ccc(Br)cc1C#N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 6/20 0.50
CYP1B1 Q16678 6/20 0.50
CYP1A2 P05177 5/20 0.50
HMGCR P04035 1/20 0.49
CYP3A4 P08684 1/20 0.49
EGFR P00533 4/20 0.41
ERBB2 P04626 3/20 0.41
NFE2L2 Q16236 2/20 0.41
ABCG2 Q9UNQ0 1/20 0.40
SRC P12931 1/20 0.40
GAK O14976 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
TSHR P16473 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
IMPDH2 P12268 1/20 0.37
IMPDH1 P20839 1/20 0.37
USP2 O75604 1/20 0.37
TNFRSF1A P19438 1/20 0.36
MEN1 O00255 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8130457 0.84 CYP1A1 (0.51) CYP1A1CYP1B1CYP1A2HMGCRCYP3A4
SCHEMBL8122560 0.82 CYP1A1 (0.50) CYP1A1CYP1B1CYP1A2HMGCRCYP3A4
SCHEMBL8124063 0.82 CYP1A1 (0.50) CYP1A1CYP1B1CYP1A2HMGCRCYP3A4
SCHEMBL8135925 0.82 CYP1A1 (0.50) CYP1A1CYP1B1CYP1A2HMGCRCYP3A4
SCHEMBL8132640 0.80 HMGCR (0.53) CYP1A1CYP1B1CYP1A2HMGCRCYP3A4
SCHEMBL7103558 0.80 CYP1A2 (0.63) CYP1A1CYP1B1CYP1A2CYP3A4NFE2L2
SCHEMBL8132635 0.80 HMGCR (0.53) CYP1A1CYP1B1CYP1A2HMGCRCYP3A4
SCHEMBL8124726 0.80 CYP1A1 (0.48) CYP1A1CYP1B1CYP1A2HMGCRCYP3A4
SCHEMBL8122816 0.79 CYP1A1 (0.47) CYP1A1CYP1B1CYP1A2HMGCRCYP3A4
SCHEMBL393816 0.76 ALDH1A1 (0.61) EGFRERBB2ALDH1A1KDM4EIMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0645382-B1 COUMARIN DERIVATIVE AND USE THEREOF MORINAGA MILK INDUSTRY CO LTD (JP) 2000-07-12 EP disclosed
EP-0645382-A1 COUMARIN DERIVATIVE AND USE THEREOF MORINAGA MILK INDUSTRY CO., LTD. (JP) 1995-03-29 EP disclosed