SCHEMBL8116655

SCHEMBL8116655

COC(=O)C(Sc1nc(OC)cc(OC)n1)C(C)(OCc1ccccc1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 12/20 0.46
EDNRA P25101 12/20 0.46
PTGES O14684 6/20 0.42
ALOX5 P09917 6/20 0.42
PPARG P37231 5/20 0.39
PSEN1 P49768 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8109239 0.84 EDNRB (0.57) EDNRBEDNRA
SCHEMBL9046722 0.82 EDNRB (0.40) EDNRBEDNRAPTGESALOX5PPARG
SCHEMBL7937196 0.82 EDNRB (0.49) EDNRBEDNRA
SCHEMBL8200442 0.80 EDNRB (0.64) EDNRBEDNRA
SCHEMBL1069539 0.79 EDNRB (0.55) EDNRBEDNRA
SCHEMBL7934306 0.76 EDNRB (0.46) EDNRBEDNRA
SCHEMBL8100747 0.75 EDNRB (0.67) EDNRBEDNRA
SCHEMBL8098308 0.75 EDNRB (0.50) EDNRBEDNRA
SCHEMBL9408612 0.74 EDNRB (0.45) EDNRBEDNRAPTGESALOX5PPARG
SCHEMBL8109266 0.73 ALDH1A1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6030975-A ANTAGONIST OF ENDOTHELINS, I.E. INHIBITION OF BINDING WITH RECEPTOR; ANTITUMOR AND -CARCINOGENIC AGENTS; SIDE EFFECT REDUCTION BASF AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed
EP-0969841-A1 USE OF CARBOXYLIC ACID DERIVATIVES FOR TREATING CANCER BASF AKTIENGESELLSCHAFT (DE) 2000-01-12 EP disclosed
WO-1998041206-A1 NOVEL CARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND USE IN TREATING CANCER BASF AKTIENGESELLSCHAFT (DE) 1998-09-24 WO disclosed
US-5703017-A HERBICIDES, PLANT GROWTH REGULATORS BASF AKTIENGESELLSCHAFT (DE) 1997-12-30 US disclosed