SCHEMBL7934306

SCHEMBL7934306

COC(=O)C(Sc1nc(C)cc(OC)n1)C(C)(c1ccccc1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 9/20 0.46
EDNRA P25101 9/20 0.46
ALDH1A1 P00352 2/20 0.43
HTT P42858 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
LMNA P02545 2/20 0.39
TSHR P16473 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7937196 0.93 EDNRB (0.49) EDNRBEDNRA
SCHEMBL7937232 0.92 KDM4E (0.44) EDNRBEDNRAALDH1A1MEN1KMT2A
SCHEMBL8098308 0.83 EDNRB (0.50) EDNRBEDNRA
SCHEMBL7928120 0.82 EDNRB (0.44) EDNRBEDNRAALDH1A1MEN1KMT2A
SCHEMBL1069539 0.80 EDNRB (0.55) EDNRBEDNRA
SCHEMBL8109239 0.79 EDNRB (0.57) EDNRBEDNRA
SCHEMBL8116655 0.76 EDNRB (0.46) EDNRBEDNRA
SCHEMBL9408612 0.70 EDNRB (0.45) EDNRBEDNRA
SCHEMBL6781616 0.70 EDNRB (0.65) EDNRBEDNRA
SCHEMBL9706660 0.69 MAPT (0.42) EDNRBEDNRAALDH1A1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235903-B1 Method for preparing sulfanyl-type endothelin receptor antagonists BASF AKTIENGESELLSCHAFT (DE) 2001-05-22 US disclosed