SCHEMBL8118487

SCHEMBL8118487

CCCCCCNCc1cccc(-c2cnc(-c3ccccc3)[nH]2)c1.Cc1ccc(CCNCc2cccc(-c3cnc(-c4ccc(F)cc4)[nH]3)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.41
CYP2D6 P10635 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP3A4 P08684 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
SCN2A Q99250 2/20 0.39
HPGDS O60760 2/20 0.39
SSTR3 P32745 4/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7141176 0.91 CYP1A2 (0.46) CYP1A2CYP2D6CYP2C19CYP3A4SCN2A
SCHEMBL7135108 0.90 CYP1A2 (0.46) CYP1A2CYP2D6CYP2C19SCN2AHPGDS
SCHEMBL8110914 0.89 CYP1A2 (0.44) CYP1A2CYP2D6CYP2C19SCN2AHPGDS
SCHEMBL7138181 0.87 HPGDS (0.49) CYP1A2CYP2D6CYP2C19CYP3A4SCN2A
SCHEMBL7143456 0.86 SCN2A (0.51) CYP1A2CYP2D6CYP2C19SCN2AHPGDS
SCHEMBL7140600 0.85 SCN2A (0.52) CYP1A2CYP2D6CYP2C19SIGMAR1SCN2A
SCHEMBL7138024 0.83 SSTR3 (0.47) SCN2AHPGDSSSTR3
SCHEMBL7143626 0.82 BACE1 (0.45) SCN2AHPGDS
SCHEMBL8189931 0.82 SCN2A (0.50) CYP1A2CYP2D6CYP2C19SCN2AHPGDS
SCHEMBL8118488 0.81 HPGDS (0.39) SCN2AHPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0996443-A1 CERTAIN DIARYLIMIDAZOLE DERIVATIVES; A NEW CLASS OF NPY SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2000-05-03 EP disclosed
WO-1999001128-A1 CERTAIN DIARYLIMIDAZOLE DERIVATIVES; A NEW CLASS OF NPY SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 1999-01-14 WO disclosed