SCHEMBL8119475

SCHEMBL8119475

COC(=O)[C@@H](CCCNC(=O)OCc1ccccc1)N=C=O

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.54
KEAP1 Q14145 2/20 0.54
NFE2L2 Q16236 2/20 0.54
LMNA P02545 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TGM2 P21980 1/20 0.49
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
FOLH1 Q04609 3/20 0.47
SLC1A3 P43003 1/20 0.46
SLC1A1 P43005 1/20 0.46
DPP8 Q6V1X1 1/20 0.46
DPP7 Q9UHL4 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8130431 0.91 HTT (0.56) HTTKEAP1NFE2L2LMNASMN1; SMN2
SCHEMBL8130436 0.91 HTT (0.56) HTTKEAP1NFE2L2LMNASMN1; SMN2
SCHEMBL8130426 0.91 HTT (0.56) HTTKEAP1NFE2L2LMNASMN1; SMN2
SCHEMBL25487774 0.81 SIRT1 (0.46)
SCHEMBL29045163 0.81 HTT (0.63) HTTKEAP1NFE2L2LMNASMN1; SMN2
SCHEMBL16574785 0.80 HTT (0.62) HTTKEAP1NFE2L2LMNASMN1; SMN2
SCHEMBL14537422 0.80 HTT (0.52) HTTKEAP1NFE2L2LMNASMN1; SMN2
SCHEMBL10705410 0.79 HTT (0.60) HTTKEAP1NFE2L2LMNASMN1; SMN2
SCHEMBL1586583 0.79 DPP8 (0.61) HTTKEAP1NFE2L2LMNASMN1; SMN2
SCHEMBL10798142 0.79 FAAH (0.46) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680469-B1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME BOEHRINGER INGELHEIM PHARMA (DE) 2000-04-26 EP disclosed