SCHEMBL8122136

SCHEMBL8122136

COc1ccc(CNC(=O)C(C)N(C(=O)Cc2ccccc2)C(=O)Cc2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.62
KMT2A Q03164 5/20 0.57
MEN1 O00255 4/20 0.57
RAB9A P51151 3/20 0.54
ALOX5 P09917 1/20 0.52
ALDH1A1 P00352 5/20 0.51
KLK7 P49862 2/20 0.51
PLA2G1B P04054 1/20 0.51
ATG4B Q9Y4P1 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
MAPT P10636 1/20 0.50
HTT P42858 1/20 0.49
KDM4E B2RXH2 1/20 0.49
CASR P41180 1/20 0.49
TSHR P16473 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5862101 0.77 NPC1 (1.00) NPC1KMT2AMEN1RAB9AALDH1A1
SCHEMBL28497417 0.77 NPC1 (1.00) NPC1KMT2AMEN1RAB9AALDH1A1
SCHEMBL4651769 0.77 NPC1 (0.49) NPC1KMT2AMEN1RAB9AALOX5
SCHEMBL16562080 0.75 NPC1 (0.77) NPC1KMT2AMEN1RAB9AALDH1A1
SCHEMBL12757447 0.75 ALDH1A1 (0.62) NPC1KMT2AMEN1RAB9AALDH1A1
SCHEMBL5017848 0.74 ALDH1A1 (0.58) NPC1KMT2AMEN1RAB9AALDH1A1
SCHEMBL16254370 0.74 NPC1 (0.60) NPC1KMT2ARAB9AALDH1A1PLA2G1B
SCHEMBL15892590 0.74 NPC1 (0.60) NPC1KMT2ARAB9AALDH1A1PLA2G1B
SCHEMBL28147642 0.74 NPC1 (0.60) NPC1KMT2ARAB9AALDH1A1PLA2G1B
SCHEMBL29699752 0.74 ALDH1A1 (0.60) NPC1KMT2AMEN1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680469-B1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME BOEHRINGER INGELHEIM PHARMA (DE) 2000-04-26 EP disclosed