SCHEMBL8123262

SCHEMBL8123262

COc1ccc(CCNC(=O)O)c(N)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 11/20 0.52
MTNR1B P49286 8/20 0.52
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
HTR2B P41595 2/20 0.47
HTR2C P28335 1/20 0.47
NQO2 P16083 3/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A1 P04798 1/20 0.46
MPO P05164 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
HTR1A P08908 1/20 0.46
CYP2D6 P10635 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
BLM P54132 1/20 0.46
PMP22 Q01453 1/20 0.46
CYP1B1 Q16678 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27002039 0.81 MTNR1A (0.66) MTNR1AMTNR1BMEN1KMT2ARAB9A
SCHEMBL8130954 0.79 MTNR1A (0.52) MTNR1AMTNR1BMEN1KMT2ANQO2
SCHEMBL4053395 0.79 POLB (0.51) MTNR1AMEN1KMT2AKDM4EALDH1A1
Hydrochloric Acid SCHEMBL5221315 0.78 HTR2A (0.52) MTNR1AMTNR1BMEN1KMT2AHTR2C
SCHEMBL5855306 0.77 ALDH1A1 (0.44) ALDH1A1RAB9A
SCHEMBL12328247 0.76 HSD17B10 (0.63) MEN1KMT2AKDM4EALDH1A1BLM
SCHEMBL3579011 0.76 ALDH1A1 (0.52) MTNR1AMEN1KMT2AKDM4EALDH1A1
SCHEMBL20957057 0.76 HSD17B10 (0.46) ALDH1A1HPGDHSD17B10
SCHEMBL4852727 0.75 ALDH1A1 (0.55) MEN1KMT2AKDM4EALDH1A1CYP3A4
SCHEMBL16428954 0.75 SMN1; SMN2 (0.44) MTNR1AMTNR1BKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526434-B1 Benzimidazolone derivatives as 5-HT1A and 5-HT2 antagonists BOEHRINGER INGELHEIM ITALIA (IT) 2000-04-19 EP disclosed
US-5576318-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS BOEHRINGER INGELHEIM ITALIA S.P.A. (IT) 1996-11-19 US disclosed
WO-1993003016-A1 BENZIMIDAZOLONE DERIVATIVES AS 5-HT1A AND 5-HT2 ANTAGONISTS BOEHRINGER INGELHEIM ITALIA S.P.A. (IT) 1993-02-18 WO disclosed
EP-0526434-A1 Benzimidazolone derivatives as 5-HT1A and 5-HT2 antagonists BOEHRINGER INGELHEIM ITALIA S.p.A. (IT) 1993-02-03 EP disclosed