SCHEMBL8124245

SCHEMBL8124245

Nc1c(Cl)cc(C=O)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
CYP3A4 P08684 1/20 0.50
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA9 Q16790 3/20 0.44
HSD17B10 Q99714 1/20 0.40
ALDH1A3 P47895 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.37
VCAM1 P19320 1/20 0.36
ALDH3A1 P30838 2/20 0.36
TDP1 Q9NUW8 2/20 0.35
POLB P06746 1/20 0.35
APEX1 P27695 1/20 0.35
HSD11B1 P28845 4/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10330733 0.86 ALDH1A1 (0.45) ALDH1A1CYP3A4CA1CA2CA9
SCHEMBL3519353 0.84 CA1 (0.50) ALDH1A1CYP3A4CA1CA2CA9
SCHEMBL1205444 0.80 ALDH1A1 (0.39) ALDH1A1CYP3A4ALDH1A3L3MBTL1POLB
SCHEMBL1312098 0.78 ALDH1A1 (0.56) ALDH1A1CYP3A4HSD17B10ALDH1A3L3MBTL1
SCHEMBL2169460 0.76 ALDH1A1 (0.54) ALDH1A1HSD17B10ALDH1A3L3MBTL1VCAM1
Fluoride SCHEMBL14358431 0.76 ALDH1A1 (0.54) ALDH1A1CYP3A4HSD17B10ALDH1A3L3MBTL1
SCHEMBL574999 0.74 ALDH1A1 (0.52) ALDH1A1CYP3A4HSD17B10
SCHEMBL8950525 0.74 ALDH1A1 (0.52) ALDH1A1HSD17B10ALDH1A3L3MBTL1VCAM1
SCHEMBL6904240 0.74 ALDH1A1 (0.52) ALDH1A1HSD17B10ALDH1A3L3MBTL1VCAM1
SCHEMBL28808069 0.74 ALDH1A1 (0.41) ALDH1A1CYP3A4HSD17B10ALDH1A3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
CN-101379111-A Polymerizable unsaturated compound and method for producing the same WAKO PURE CHEM IND LTD (JP) 2009-03-04 CN disclosed
EP-0680469-B1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME BOEHRINGER INGELHEIM PHARMA (DE) 2000-04-26 EP disclosed
US-5807875-A OBESITY THERAPY DR. KARL THOMAE GMBH (DE) 1998-09-15 US disclosed
US-5616620-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-04-01 US disclosed
EP-0680469-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME Dr. Karl Thomae GmbH (DE) 1995-11-08 EP disclosed
WO-1994017035-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME DR. KARL THOMAE GMBH (DE) 1994-08-04 WO disclosed
US-5216170-A Promoters of livestock; treatment of obesity BAYER AKTIENGESELLSCHAFT (DE) 1993-06-01 US disclosed
US-5028617-A Heteroarylethanol-pyridylalkylamines for controlling animal growth BAYER AKTIENGESELLSCHAFT (DE) 1991-07-02 US disclosed
EP-0379928-A2 Aryl- and heteroarylethanol-pyridylalkylamines, process for their preparation and their use as performance stimulators by animals and as anti-adipositas agent BAYER AG (DE) 1990-08-01 EP disclosed
US-4678797-A INSECTICIDES, MITICIDES, NEMATOCIDES, FUNGICIDES, FEED UTILIZATION BAYER AKTIENGESELLSCHAFT (DE) 1987-07-07 US disclosed
EP-0162383-A1 Biologically active agent containing substituted isoxazolidines, isoxazolidines and their preparation BAYER AG (DE) 1985-11-27 EP disclosed
US-4087528-A POTENTIATORS OF ANTIBACTERIAL SULFA DRUGS ABBOTT LABORATORIES (US) 1978-05-02 US disclosed
US-4008236-A 2,4-Diamino-5-benzylpyrimidines ABBOTT LABORATORIES (US) 1977-02-15 US disclosed