SCHEMBL8124408

SCHEMBL8124408

O=C(c1cccc([N+](=O)[O-])c1)c1ccc(Cl)cc1[N+](=O)[O-]

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
TSHR P16473 2/20 0.55
CES2 O00748 2/20 0.54
CES1 P23141 1/20 0.54
TDP1 Q9NUW8 1/20 0.53
TP53 P04637 1/20 0.53
LMNA P02545 5/20 0.48
HTT P42858 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
F2 P00734 1/20 0.48
PLAU P00749 1/20 0.48
KLKB1 P03952 1/20 0.48
ELANE P08246 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
HPGD P15428 1/20 0.48
CYP2C19 P33261 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11289155 0.85 HPGD (0.59) ALDH1A1CES2LMNAL3MBTL1SMN1; SMN2
SCHEMBL9422048 0.84 ALDH1A1 (0.56) ALDH1A1TSHRCES2CES1TDP1
SCHEMBL11507878 0.84 ALDH1A1 (0.56) ALDH1A1TSHRCES2CES1TDP1
SCHEMBL10341585 0.82 CES2 (0.60) ALDH1A1TSHRCES2CES1TP53
SCHEMBL14984180 0.82 ALDH1A1 (0.68) ALDH1A1TSHRCES2CES1TDP1
SCHEMBL11301098 0.82 HPGD (0.59) ALDH1A1TSHRHTTSMN1; SMN2CYP1A2
SCHEMBL10903202 0.82 ALDH1A1 (0.56) ALDH1A1TSHRCES2CES1TDP1
SCHEMBL10902732 0.81 MAPK1 (0.63) ALDH1A1TSHRCES2CES1TDP1
SCHEMBL7787760 0.81 ALDH1A1 (0.63) ALDH1A1TSHRCES2CES1TDP1
SCHEMBL8962890 0.80 CES2 (0.57) ALDH1A1TSHRCES2CES1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973777-A1 FUROPYRIDINE, THIENOPYRIDINE, PYRROLOPYRIDINE AND RELATED PYRIMIDINE, PYRIDAZINE AND TRIAZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-01-26 EP disclosed
US-6001849-A Furopyridine, thienopyridine pyrrolopyridine useful in controlling chemical synaptic transmission ABBOTT LABORATORIES (US) 1999-12-14 US disclosed
EP-0934308-A1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 1999-08-11 EP disclosed
WO-1998046609-A1 FUROPYRIDINE, THIENOPYRIDINE, PYRROLOPYRIDINE AND RELATED PYRIMIDINE, PYRIDAZINE AND TRIAZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1998-10-22 WO disclosed
WO-1997046554-A1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1997-12-11 WO disclosed