SCHEMBL8124648

SCHEMBL8124648

CCN(CC)CC(O)Cn1c2ccccc2c2c3c(c4c5ccccc5[nH]c4c21)C(=O)NC3=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKD3 O94806 5/20 0.68
PRKCG P05129 5/20 0.68
PRKCB P05771 5/20 0.68
PRKCA P17252 5/20 0.68
PRKCH P24723 5/20 0.68
PRKCI P41743 5/20 0.68
PRKCE Q02156 5/20 0.68
PRKCQ Q04759 5/20 0.68
PRKCZ Q05513 5/20 0.68
PRKCD Q05655 5/20 0.68
PRKD1 Q15139 5/20 0.68
CDK4 P11802 9/20 0.61
CCND1 P24385 9/20 0.61
CCNE2 O96020 4/20 0.61
CCNE1 P24864 4/20 0.61
CDK2 P24941 4/20 0.61
PRKACA P17612 4/20 0.60
PRKACG P22612 4/20 0.60
PRKACB P22694 4/20 0.60
MYLK Q15746 3/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8127615 0.90 PRKCA (0.54) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL9197404 0.87 MYLK (0.62) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL9204314 0.87 MYLK (0.63) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL8113741 0.86 CDK4 (0.70) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL8113301 0.85 MYLK (0.81) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL8316417 0.81 PRKD3 (1.00) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL13075769 0.79 CDK4 (0.79) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL9834250 0.76 TSHR (0.57) CDK4CCND1PRKACAPRKACGPRKACB
SCHEMBL8463787 0.75 CDK4 (1.00) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL8120626 0.75 CDK4 (0.80) PRKD3PRKCGPRKCBPRKCAPRKCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0642513-B1 INDOLOCARBAZOLE IMIDES AND THEIR USE KTB TUMORFORSCHUNGSGESELLSCHAF (DE) 2000-08-09 EP claimed
US-5883114-A TREATING CANCEROUS TUMORS, INFLAMMATORY DISEASES, AND ALLERGIES GOEDECKE AKTIENGESELLSCHAFT (DE) 1999-03-16 US claimed
EP-0642513-A1 INDOLOCARBAZOLE IMIDES AND THEIR USE GÖDECKE AKTIENGESELLSCHAFT (DE) 1995-03-15 EP claimed
WO-1993024491-A1 INDOLOCARBAZOLE IMIDES AND THEIR USE Gödecke Aktiengesellschaft (DE) 1993-12-09 WO claimed
EP-0642513-B1 INDOLOCARBAZOLE IMIDES AND THEIR USE KTB TUMORFORSCHUNGSGESELLSCHAF (DE) 2000-08-09 EP disclosed
US-5945440-A Indolocarbazole imides and the use thereof GOEDECKE AKTIENGESELLSCHAFT (DE) 1999-08-31 US disclosed
US-5883114-A TREATING CANCEROUS TUMORS, INFLAMMATORY DISEASES, AND ALLERGIES GOEDECKE AKTIENGESELLSCHAFT (DE) 1999-03-16 US disclosed
EP-0642513-A1 INDOLOCARBAZOLE IMIDES AND THEIR USE GÖDECKE AKTIENGESELLSCHAFT (DE) 1995-03-15 EP disclosed
WO-1993024491-A1 INDOLOCARBAZOLE IMIDES AND THEIR USE Gödecke Aktiengesellschaft (DE) 1993-12-09 WO disclosed