SCHEMBL8125239

SCHEMBL8125239

ICCc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 15/20 0.49
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
ENPP2 Q13822 1/20 0.37
ALOX15 P16050 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
ALOX12 P18054 1/20 0.35
CASP1 P29466 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NMBR P28336 1/20 0.33
MEN1 O00255 1/20 0.31
SLC22A1 O15245 1/20 0.31
KCNN4 O15554 1/20 0.31
NR1I2 O75469 1/20 0.31
GMNN O75496 1/20 0.31
USP2 O75604 1/20 0.31
TRPM2 O94759 1/20 0.31
ABCB11 O95342 1/20 0.31
EGFR P00533 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6345609 0.87 SIRT2 (0.45) SIRT2CYP11B1CYP11B2ENPP2ALOX15
SCHEMBL1041048 0.84 SIRT2 (0.49) SIRT2CYP11B1CYP11B2ENPP2NMBR
SCHEMBL2035093 0.84 SIRT2 (0.49) SIRT2CYP11B1CYP11B2ENPP2CYP2C9
SCHEMBL7159342 0.84 SIRT2 (0.49) SIRT2CYP11B1CYP11B2ENPP2ALOX15
SCHEMBL14993551 0.84 SIRT2 (0.49) SIRT2CYP11B1CYP11B2ENPP2ALOX15
SCHEMBL4382643 0.84 SIRT2 (0.54) SIRT2CYP11B1CYP11B2ENPP2CYP19A1
SCHEMBL8794940 0.84 SIRT2 (0.49) SIRT2CYP11B1CYP11B2ENPP2ALOX15
SCHEMBL7988316 0.83 SIRT2 (0.48) SIRT2CYP11B1CYP11B2ENPP2ALOX15
Hydrochloric Acid SCHEMBL7987252 0.83 SIRT2 (0.53) SIRT2CYP11B1CYP11B2ENPP2CYP19A1
SCHEMBL2490264 0.83 SIRT2 (0.48) SIRT2CYP11B1CYP11B2ENPP2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016514-A2 1, 3 AND 1, 3, 5 SUBSTITUTED IMIDAZOLES AS ANTIHYPERTENSIVA ELDRUG S.A. (GR) 2009-02-05 WO disclosed