SCHEMBL8125702

SCHEMBL8125702

Cc1ccc(C2CC(c3cc[nH]c3C)CCN2)cc1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PRCP P42785 1/20 0.33
MAPT P10636 1/20 0.33
GID4 Q8IVV7 1/20 0.33
MKNK1 Q9BUB5 1/20 0.32
GFER P55789 1/20 0.31
KDM1A O60341 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8131062 0.89 HTR3A (0.39) PRCPMKNK1KDM1A
SCHEMBL8125194 0.89 SLC6A2 (0.32) PRCPMKNK1
SCHEMBL8115602 0.89 SLC18A3 (0.38) PRCP
SCHEMBL8124405 0.87 MKNK1 (0.34) MKNK1KDM1A
SCHEMBL8125817 0.83 KDM1A (0.34) KDM1A
SCHEMBL8131566 0.83 SLC6A2 (0.38) MAPT
SCHEMBL8128593 0.82 SLC6A4 (0.36) KDM1A
SCHEMBL8115493 0.81
SCHEMBL8124867 0.79 SLC6A2 (0.36) GID4
SCHEMBL8124794 0.79 SLC6A2 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054887-A1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS Amgen Inc. (US) 2000-11-29 EP claimed
WO-1999040091-A1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS AMGEN INC. (US) 1999-08-12 WO claimed
EP-1054887-A1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS Amgen Inc. (US) 2000-11-29 EP disclosed
WO-1999040091-A1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS AMGEN INC. (US) 1999-08-12 WO disclosed