SCHEMBL8127237

SCHEMBL8127237

CN1CCc2ccc(NC(=O)Nc3ccc(F)c(Cl)c3)cc2C1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.57
MEN1 O00255 7/20 0.56
KMT2A Q03164 7/20 0.56
HTT P42858 3/20 0.56
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
LMNA P02545 2/20 0.56
MAPT P10636 5/20 0.53
DRD2 P14416 1/20 0.53
HTR2A P28223 1/20 0.53
HTR2C P28335 1/20 0.53
DRD3 P35462 1/20 0.53
HTR6 P50406 1/20 0.53
CASP3 P42574 1/20 0.52
SENP7 Q9BQF6 1/20 0.52
ALDH1A1 P00352 1/20 0.51
MCHR1 Q99705 2/20 0.51
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8116428 0.89 LMNA (0.53) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL8131703 0.85 RAB9A (0.66) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL8128776 0.84 MAPT (0.60) MEN1KMT2AHTTNPC1RAB9A
SCHEMBL8132295 0.83 MAPT (0.54) SLC2A1MEN1KMT2AHTTNPC1
SCHEMBL6293985 0.82 NPC1 (0.50) HTTNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL8161154 0.82 NPC1 (0.70) MEN1KMT2AHTTNPC1RAB9A
SCHEMBL8126912 0.81 RAB9A (0.68) MEN1KMT2AHTTNPC1RAB9A
SCHEMBL8130701 0.81 NPC1 (0.65) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL8124101 0.80 NPC1 (0.57) MEN1KMT2ANPC1RAB9ALMNA
SCHEMBL8135393 0.79 EPHX2 (0.59) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1005459-A1 SUBSTITUTED ISOQUINOLINES AS ANTICONVULSIVANTS SMITHKLINE BEECHAM PLC (GB) 2000-06-07 EP disclosed
WO-1999014197-A1 SUBSTITUTED ISOQUINOLINES AS ANTICONVULSIVANTS SMITHKLINE BEECHAM PLC (GB) 1999-03-25 WO disclosed