SCHEMBL8129124

SCHEMBL8129124

CCCCC(CC(=O)O)c1ccc(OCc2ccccc2)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 5/20 0.51
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.42
MMP12 P39900 1/20 0.42
PTGES O14684 1/20 0.42
ALOX5 P09917 1/20 0.42
PPARG P37231 1/20 0.42
MAOB P27338 1/20 0.42
GSK3B P49841 1/20 0.41
CTRC Q99895 1/20 0.41
MTNR1A P48039 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8136349 0.97 FFAR1 (0.50) FFAR1KMT2ASMN1; SMN2L3MBTL1MMP12
SCHEMBL8121730 0.89 FFAR1 (0.51) FFAR1MAOB
SCHEMBL8132546 0.86 HDAC3 (0.44) FFAR1ALOX5PPARG
SCHEMBL8120029 0.85 FFAR1 (0.47) FFAR1KMT2ASMN1; SMN2
SCHEMBL8121726 0.85 FFAR1 (0.48) FFAR1MAOB
SCHEMBL8136073 0.84 PPARG (0.43) FFAR1PTGESALOX5PPARG
SCHEMBL8119916 0.83 CYSLTR2 (0.45) FFAR1
SCHEMBL8126572 0.82 CYSLTR2 (0.47) FFAR1
SCHEMBL8130408 0.81 THRA (0.43) FFAR1PTGESALOX5PPARG
SCHEMBL8129412 0.80 FFAR1 (0.40) FFAR1SMN1; SMN2PTGESALOX5PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0763524-B1 Urea and amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prophylactic use SANKYO CO (JP) 2000-08-23 EP disclosed
US-6040339-A TREATMENT AND PROPHYLAXIS OF HYPERCHOLESTEREMIA OR ARTERIOSCLEROSIS IN A MAMMAL SANKYO COMPANY, LIMITED (JP) 2000-03-21 US disclosed
US-5880147-A Amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prohylactic use SANKYO COMPANY, LIMITED (JP) 1999-03-09 US disclosed
EP-0763524-A1 Urea and amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prophylactic use SANKYO COMPANY LIMITED (JP) 1997-03-19 EP disclosed