SCHEMBL8129204

SCHEMBL8129204

CC1CCC(=O)c2cc(Br)ccc2S1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 1/20 0.41
KLK7 P49862 1/20 0.41
PBRM1 Q86U86 1/20 0.41
S100A4 P26447 1/20 0.35
PARP10 Q53GL7 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
VHL P40337 1/20 0.34
ELOC Q15369 1/20 0.34
ELOB Q15370 1/20 0.34
PARP1 P09874 1/20 0.34
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
PTPRC P08575 1/20 0.32
MAOB P27338 2/20 0.32
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8110022 0.84 KDM4E (0.54) KDM4EALDH1A1HPGDKLK7PBRM1
SCHEMBL18753241 0.81 KDM4E (0.41) KDM4EALDH1A1HPGDKLK7VHL
SCHEMBL13043709 0.81 VHL (0.55) KDM4EALDH1A1HPGDKLK7S100A4
SCHEMBL7418018 0.77 PNMT (0.38) PARP10PARP11HTR2AHTR2C
SCHEMBL9367610 0.73 HTR2A (0.39) PARP10TDP1L3MBTL1PARP1HTR2A
SCHEMBL13497572 0.73 VHL (0.53) KDM4EALDH1A1HPGDKLK7S100A4
SCHEMBL30917697 0.72 PBRM1 (0.44) PBRM1S100A4PARP10TDP1L3MBTL1
SCHEMBL30917701 0.72 PBRM1 (0.44) PBRM1S100A4PARP10TDP1L3MBTL1
SCHEMBL8617679 0.72 PBRM1 (0.44) PBRM1S100A4PARP10TDP1L3MBTL1
SCHEMBL31650648 0.72 PBRM1 (0.44) PBRM1S100A4PARP10TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1039899-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
WO-1999032100-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed