SCHEMBL8129247

SCHEMBL8129247

CCCCCC(CC(=O)Nc1cc(C(N)=O)ccc1C(C)(C)C)c1ccc(OC(C)C)cc1OC

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 4/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 4/20 0.38
LMNA P02545 3/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 1/20 0.37
LPAR1 Q92633 1/20 0.36
PARP10 Q53GL7 1/20 0.35
MAPK1 P28482 2/20 0.34
HTT P42858 1/20 0.34
GAA P10253 2/20 0.33
XBP1 P17861 1/20 0.33
ATM Q13315 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ERAP2 Q6P179 1/20 0.33
LNPEP Q9UIQ6 1/20 0.33
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8119996 0.94 LPAR1 (0.41) L3MBTL1KMT2AALDH1A1MAPTLPAR1
SCHEMBL8131084 0.93 LPAR1 (0.41) L3MBTL1KMT2AALDH1A1MAPTLPAR1
SCHEMBL8128380 0.93 KMT2A (0.39) L3MBTL1KMT2AALDH1A1LMNAHPGD
SCHEMBL8121344 0.92 LPAR1 (0.42) L3MBTL1KMT2AALDH1A1MAPTLPAR1
SCHEMBL8148224 0.91 ALDH1A1 (0.38) L3MBTL1ALDH1A1LMNAHPGDMAPT
SCHEMBL8129418 0.90 KMT2A (0.37) L3MBTL1KMT2AALDH1A1LPAR1MAPK1
SCHEMBL8129485 0.90 MAPK1 (0.38) L3MBTL1KMT2ALPAR1MAPK1
SCHEMBL8120272 0.89 KMT2A (0.39) L3MBTL1KMT2ALMNAHPGDMAPK1
SCHEMBL8128937 0.89 KMT2A (0.40) L3MBTL1KMT2AMAPK1
SCHEMBL8129666 0.89 L3MBTL1 (0.42) L3MBTL1KMT2AALDH1A1MAPTLPAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0763524-B1 Urea and amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prophylactic use SANKYO CO (JP) 2000-08-23 EP disclosed
US-6040339-A TREATMENT AND PROPHYLAXIS OF HYPERCHOLESTEREMIA OR ARTERIOSCLEROSIS IN A MAMMAL SANKYO COMPANY, LIMITED (JP) 2000-03-21 US disclosed
US-5880147-A Amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prohylactic use SANKYO COMPANY, LIMITED (JP) 1999-03-09 US disclosed
EP-0763524-A1 Urea and amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prophylactic use SANKYO COMPANY LIMITED (JP) 1997-03-19 EP disclosed