SCHEMBL8129263

SCHEMBL8129263

O=CCC1(c2ccc(Cl)cc2)CCN(C(=O)c2ccccc2)C1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.48
CHRM3 P20309 3/20 0.48
ALDH1A1 P00352 2/20 0.47
LMNA P02545 2/20 0.47
TACR2 P21452 3/20 0.46
TACR1 P25103 2/20 0.46
MGLL Q99685 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
RIPK1 Q13546 1/20 0.44
CCR8 P51685 1/20 0.43
KCNH2 Q12809 1/20 0.43
CCR1 P32246 1/20 0.43
KCNA5 P22460 1/20 0.43
DDB1 Q16531 2/20 0.43
CRBN Q96SW2 2/20 0.43
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8143470 0.93 EPHX2 (0.50) CHRM2CHRM3ALDH1A1LMNATACR2
SCHEMBL8143466 0.93 EPHX2 (0.50) CHRM2CHRM3ALDH1A1LMNATACR2
SCHEMBL6947952 0.87 TACR2 (0.61) TACR2TACR1
SCHEMBL3523461 0.84 CCR5 (0.51) CHRM2CHRM3ALDH1A1LMNARIPK1
SCHEMBL8119487 0.84 EPHX2 (0.57) CHRM2CHRM3ALDH1A1LMNATACR2
SCHEMBL8148884 0.81 TACR2 (0.60) TACR2TACR1
SCHEMBL8148888 0.81 TACR2 (0.60) TACR2TACR1
SCHEMBL8150748 0.80 TACR2 (0.46) ALDH1A1TACR2TACR1
SCHEMBL8150747 0.80 TACR2 (0.46) ALDH1A1TACR2TACR1
SCHEMBL6998425 0.76 EPHX2 (0.53) CHRM2CHRM3ALDH1A1LMNATACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0992493-A1 Substituted benzoylpiperidine derivatives and their use as Neurokinin antagonists PFIZER INC. (US) 2000-04-12 EP disclosed