SCHEMBL8129369

SCHEMBL8129369

CC(C)COC(=O)CC1(O)CCC(N2CCNCC2)CC1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.33
KCNH2 Q12809 1/20 0.32
GRIN2B Q13224 1/20 0.32
CYP2C19 P33261 1/20 0.31
PADI1 Q9ULC6 1/20 0.31
PADI4 Q9UM07 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7300028 0.80 CYP2C19 (0.33) KCNH2GRIN2BCYP2C19HRH3
SCHEMBL19625756 0.68 HPGD (0.40) HRH3
SCHEMBL21946897 0.68 CHRM5 (0.51) RAB9APADI1PADI4
SCHEMBL8184493 0.67 KCNH2 (0.39) KCNH2GRIN2B
SCHEMBL20179968 0.66 CHRM5 (0.50) RAB9APADI1PADI4
SCHEMBL21695211 0.66 CHRM5 (0.50) RAB9APADI1PADI4
SCHEMBL9052473 0.66 OPRM1 (0.38)
SCHEMBL19450983 0.65 CHRM5 (0.41) RAB9APADI1PADI4
SCHEMBL27510467 0.65 HRH3 (0.33) HRH3
SCHEMBL27295498 0.65 SLC6A1 (0.38) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0895475-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2000-08-23 EP disclosed
EP-0895475-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-02-10 EP disclosed
WO-1997024122-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed