SCHEMBL8130601

SCHEMBL8130601

CCN(CCN(CCN(CC(=O)O)CC(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)CC(=O)OC(C)(C)C)CC(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.36
CHRM2 P08172 2/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
ADRA2A P08913 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
DRD1 P21728 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
CYP2C19 P33261 1/20 0.36
ADRA1A P35348 1/20 0.36
DRD3 P35462 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
SLC6A3 Q01959 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
EYA2 O00167 1/20 0.33
APP P05067 1/20 0.33
ACE P12821 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8135274 0.99 TDP1 (0.34) TDP1CHRM2KDM4ELMNAADRA2A
SCHEMBL7203307 0.92 CHRM2 (0.33) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL7762658 0.88 CHRM2 (0.32) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL7129262 0.87 TDP1 (0.47) TDP1CHRM2KDM4ELMNAADRA2A
SCHEMBL5555346 0.84
SCHEMBL8132756 0.83 SYK (0.40) CHRM2TSHRCHRM4CHRM5CHRM1
SCHEMBL8875240 0.82 AKT1 (0.40) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL8120285 0.82 AKT1 (0.40) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL8134806 0.81 SYK (0.40) CHRM2TSHRCHRM4CHRM5CHRM1
SCHEMBL8137127 0.81 AKT1 (0.40) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080785-A REACTING A ALKYLNEDI-PRIMARY AMINE COMPOUND WITH A PROTECTIVE GROUP SUCH AS TRIFLUOROACETYL OR BENZYL GROUP REAGENT TO FORM AN INTERMEDIATE, REACTING THE INTERMEDIATE WITH HALOACETIC TERT-BYTYL ESTER TO FORM ESTER GROUPS, DEPROTECTING SCHERING AKTIENGESELLSCHAFT (DE) 2000-06-27 US disclosed