SCHEMBL8135451

SCHEMBL8135451

B(c1ccccc1)c1ccccc1.OC[C@@H]1CCCN1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
LTA4H P09960 5/20 0.42
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
HTR6 P50406 4/20 0.40
GHSR Q92847 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Biphenyl SCHEMBL5439264 0.84 POLB (0.51) POLBLTA4HCHRNB4CHRNA3HTR6
Biphenyl SCHEMBL4430290 0.84 POLB (0.51) POLBLTA4HCHRNB4CHRNA3HTR6
SCHEMBL9015256 0.81 POLB (0.57) POLBLTA4H
SCHEMBL10141198 0.78
SCHEMBL115932 0.78
SCHEMBL10141207 0.78
SCHEMBL145266 0.78
SCHEMBL19071 0.78
SCHEMBL7787365 0.78 FDPS (0.41) POLBCHRNB4CHRNA3GHSR
Hydrochloric Acid SCHEMBL4742761 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668266-B1 Process for preparing 1,1-diarylprolinols MERCK & CO INC (US) 2000-02-02 EP disclosed
EP-0962451-A2 Chiral catalysts for reduction of ketones and process for their preparation MERCK & CO. INC. (US) 1999-12-08 EP disclosed
EP-0453298-B1 Chiral catalysts for reduction of ketones and process for their preparation MERCK & CO INC (US) 1995-12-06 EP disclosed
US-5189177-A Chiral boron catalysts for reduction of ketones and process for their preparation MERCK & CO., INC. (US) 1993-02-23 US disclosed
EP-0453298-A2 Chiral catalysts for reduction of ketones and process for their preparation MERCK & CO. INC. (US) 1991-10-23 EP disclosed
US-5039802-A Arylation process for preparation of chiral catalysts for ketone reduction MERCK & CO., INC. (US) 1991-08-13 US disclosed