SCHEMBL8136123

SCHEMBL8136123

CCOC(=O)C(C(=O)OCC)C(=O)c1cc(Cl)c(Cl)cc1[N+](=O)[O-]

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.41
LMNA P02545 4/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 2/20 0.41
GALR2 O43603 1/20 0.41
MITF O75030 1/20 0.41
HSP90AA1 P07900 1/20 0.41
XBP1 P17861 1/20 0.41
CCR6 P51684 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
THRB P10828 1/20 0.40
HPD P32754 1/20 0.39
VCAM1 P19320 1/20 0.38
MAPT P10636 2/20 0.38
PDK1 Q15118 1/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPC1 O15118 1/20 0.38
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8136193 0.92 RECQL (0.44) POLBLMNAALDH1A1HPGDGALR2
SCHEMBL8139201 0.84 HPGD (0.53) POLBALDH1A1HPGDSMN1; SMN2HPD
SCHEMBL10803120 0.80 MAPT (0.42) POLBLMNAALDH1A1HPGDGALR2
SCHEMBL13312378 0.78 HPD (0.46) POLBLMNAALDH1A1HPGDGALR2
SCHEMBL9860199 0.78 ALDH1A1 (0.44) POLBLMNAALDH1A1HPGDGALR2
SCHEMBL8144060 0.77 MAPT (0.55) LMNAALDH1A1SMN1; SMN2HPDMAPT
SCHEMBL8137056 0.77 ALDH1A1 (0.55) LMNAALDH1A1HPGDSMN1; SMN2NPSR1
SCHEMBL8489229 0.76 HPD (0.69) LMNAALDH1A1THRBHPDMAPT
SCHEMBL27474538 0.75 ALDH1A1 (0.53) POLBLMNAALDH1A1HPGDGALR2
SCHEMBL6406686 0.75 TSHR (0.57) POLBLMNAALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760819-B1 TRICYCLIC DICARBONYL DERIVATIVES HOFFMANN LA ROCHE (CH) 2000-07-19 EP disclosed
US-5688803-A BRAIN DISORDERS; PSYCHOLOGICAL DISORDERS HOFFMANN-LA ROCHE INC. (US) 1997-11-18 US disclosed
EP-0760819-A1 TRICYCLIC DICARBONYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed
WO-1995032205-A1 TRICYCLIC DICARBONYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1995-11-30 WO disclosed