SCHEMBL8136163

SCHEMBL8136163

CCOC(=O)c1ccc(-c2ccc(N)c3c2CCN(C)C3)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.49
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 3/20 0.49
HSD17B10 Q99714 2/20 0.49
POLB P06746 1/20 0.49
ALOX15 P16050 1/20 0.49
CYP1A2 P05177 2/20 0.45
LMNA P02545 1/20 0.45
CYP3A4 P08684 1/20 0.45
MAOA P21397 1/20 0.45
CYP2C9 P11712 2/20 0.43
FDFT1 P37268 1/20 0.42
KCNH2 Q12809 2/20 0.42
HRH3 Q9Y5N1 1/20 0.42
VDR P11473 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8137079 0.83 ALDH1A1 (0.48) MAPK1KDM4EALDH1A1HSD17B10POLB
SCHEMBL8140152 0.77 ALDH1A1 (0.49) MAPK1KDM4EALDH1A1HSD17B10POLB
SCHEMBL8133556 0.76 MAPK1 (0.46) MAPK1KDM4EALDH1A1HSD17B10POLB
SCHEMBL5102962 0.76 MAPK1 (0.46) MAPK1KDM4EALDH1A1HSD17B10POLB
SCHEMBL5102959 0.76 MAPK1 (0.46) MAPK1KDM4EALDH1A1HSD17B10POLB
SCHEMBL6611465 0.75 HDAC1 (0.38)
SCHEMBL13592435 0.75 GRIA1 (0.34) KDM4EALDH1A1CYP1A2MAOAKCNH2
SCHEMBL14287214 0.74 LMNA (0.50) MAPK1KDM4EALDH1A1HSD17B10LMNA
Hydrochloric Acid SCHEMBL4377355 0.74 MEN1 (0.41) POLBCYP1A2CYP3A4MAOACYP2C9
Hydrochloric Acid SCHEMBL6613546 0.73 ALDH1A1 (0.42) MAPK1KDM4EALDH1A1CYP1A2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0781285-B1 FUSED INDOLE AND QUINOXALINE DERIVATIVES, THEIR PREPARATION AND USE AS GLUTAMATE ANTAGONISTS NEUROSEARCH AS (DK) 2000-01-12 EP disclosed
US-5801174-A CEREBROVASCULAR DISORDERS NEUROSEARCH A/S (DK) 1998-09-01 US disclosed