SCHEMBL8136527

SCHEMBL8136527

CSc1ccnc(SCc2ccc3c(c2)CCO3)n1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LYPLAL1 Q5VWZ2 1/20 0.43
GSK3B P49841 12/20 0.41
TP53 P04637 1/20 0.40
KDM4E B2RXH2 1/20 0.38
MET P08581 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8178419 0.82 DYRK1A (0.46) LYPLAL1GSK3BTP53
SCHEMBL12204567 0.74 GSK3B (0.57) LYPLAL1GSK3BKDM4E
SCHEMBL13461945 0.73 RAB9A (0.46) GSK3B
SCHEMBL6636334 0.71 LYPLAL1 (0.50) LYPLAL1GSK3BTP53KDM4E
SCHEMBL27545516 0.71 MEN1 (0.44)
SCHEMBL30965 0.67 KDM4E (0.51) KDM4E
SCHEMBL3491505 0.65 GSK3B (0.83) GSK3B
SCHEMBL22766338 0.65 PRKCI (0.49) TP53KDM4E
SCHEMBL31248520 0.65 GSK3B (0.58) GSK3B
SCHEMBL14486664 0.64 DAO (0.58) GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1034167-A1 ALPHA-ALKYLTHIO SUBSTITUTED PYRIMIDINE ETHERS AND THIOETHERS AS VIRAL REVERSE TRANSCRIPTASE INHIBITORS PHARMACIA & UPJOHN COMPANY (US) 2000-09-13 EP disclosed
WO-1999019304-A2 ALPHA-ALKYLTHIO SUBSTITUTED PYRIMIDINE ETHERS AND THIOETHERS AS VIRAL REVERSE TRANSCRIPTASE INHIBITORS PHARMACIA & UPJOHN COMPANY (US) 1999-04-22 WO disclosed