SCHEMBL8137182

SCHEMBL8137182

Nc1ccc(-c2ncc[nH]2)cc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.53
MTOR P42345 1/20 0.52
ADK P55263 1/20 0.52
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
CYP19A1 P11511 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
SMPD3 Q9NY59 1/20 0.41
ADRA2A P08913 3/20 0.40
CYP17A1 P05093 1/20 0.40
CYP11B1 P15538 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8536727 0.84 ALDH1A1 (0.52) NISCHMTORADKMEN1KMT2A
SCHEMBL3649556 0.84 NISCH (0.58) NISCHMTORADKTDP1ALDH1A1
SCHEMBL1838153 0.84 NISCH (0.58) NISCHMTORADKTDP1ALDH1A1
SCHEMBL7060159 0.84 NISCH (0.49) NISCHMTORADKMEN1KMT2A
Hydrochloric Acid SCHEMBL27817951 0.82 NISCH (0.56) NISCHMTORADKTDP1ALDH1A1
Hydrochloric Acid SCHEMBL3646836 0.82 NISCH (0.56) NISCHMTORADKTDP1ALDH1A1
SCHEMBL12714764 0.80 SMPD3 (0.60) NISCHMTORADKMEN1KMT2A
SCHEMBL7425938 0.80 NISCH (0.45) NISCHMTORADKALDH1A1KDM4E
SCHEMBL27963202 0.80 SMPD3 (0.56) NISCHMTORADKMEN1KMT2A
SCHEMBL722191 0.79 NISCH (0.78) NISCHMTORADKMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0556393-B1 FUSED PYRAZINE DERIVATIVE YAMANOUCHI PHARMA CO LTD (JP) 2000-07-26 EP disclosed
WO-1996040997-A1 METHOD OF FLUORESCENT DETECTION OF NUCLEIC ACIDS AND CYTOSKELETON ELEMENTS USING BIS-DICATIONIC ARYL FURANS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-12-19 WO disclosed
US-5283244-A Anticonvulsants, nervous system disorders YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-02-01 US disclosed
EP-0556393-A1 FUSED PYRAZINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1993-08-25 EP disclosed