SCHEMBL7425938

SCHEMBL7425938

N#Cc1cc(-c2ncc[nH]2)ccc1N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.45
MTOR P42345 1/20 0.43
ADK P55263 1/20 0.43
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
CHEK1 O14757 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP19A1 P11511 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
TBK1 Q9UHD2 1/20 0.38
PRKACA P17612 2/20 0.37
PRKACG P22612 2/20 0.37
PRKACB P22694 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8137182 0.80 NISCH (0.53) NISCHMTORADKKDM4EALDH1A1
SCHEMBL8538740 0.79 NISCH (0.46) NISCHMTORADKKDM4EALDH1A1
SCHEMBL8537240 0.78 CYP11B2 (0.48) NISCH
SCHEMBL3978330 0.78 NISCH (0.45) NISCHMTORADKKDM4EALDH1A1
SCHEMBL8539165 0.76 MAPT (0.40) NISCHMTORADKKDM4EALDH1A1
SCHEMBL8536727 0.76 ALDH1A1 (0.52) NISCHMTORADKKDM4EALDH1A1
SCHEMBL1838153 0.76 NISCH (0.58) NISCHMTORADKKDM4EALDH1A1
SCHEMBL7060159 0.76 NISCH (0.49) NISCHMTORADKKDM4EALDH1A1
SCHEMBL5072719 0.75 TDP1 (0.48) KDM4EALDH1A1CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL27817951 0.74 NISCH (0.56) NISCHMTORADKKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691967-A1 NITROGEN-CONTAINING FUSED-HETEROCYCLE COMPOUNDS Eisai Co., Ltd. (JP) 1996-01-17 EP disclosed
WO-1994022855-A1 NITROGEN-CONTAINING FUSED-HETEROCYCLE COMPOUNDS EISAI CO., LTD. (JP) 1994-10-13 WO disclosed