SCHEMBL8137658

SCHEMBL8137658

COC(=O)Nc1cccc(C)c1COc1cccn2c(C=O)c(C)nc12

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
GUCY1B2 O75343 10/20 0.45
GUCY1A2 P33402 10/20 0.45
GUCY1A1 Q02108 10/20 0.45
GUCY1B1 Q02153 10/20 0.45
BDKRB2 P30411 1/20 0.43
ATP4A P20648 1/20 0.43
ATP4B P51164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7839635 0.92 CYP1A2 (0.49) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7505990 0.92 CYP1A2 (0.51) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7499698 0.90 CYP1A2 (0.49) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8805202 0.90 CYP1A2 (0.53) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1817623 0.88 CYP3A4 (0.73) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9097105 0.87 CYP1A2 (0.58) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1814241 0.86 ATP4A (0.60) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8136776 0.84 CYP3A4 (0.53) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9685702 0.83 CYP1A2 (0.53) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7499038 0.83 CYP3A4 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683780-B1 IMIDAZOPYRIDINES AND THEIR USE IN TREATING GASTROINTESTINAL DISEASES BYK GULDEN LOMBERG CHEM FAB (DE) 2000-04-26 EP disclosed
US-5665730-A GASTROINTESTINAL DISORDERS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1997-09-09 US disclosed