SCHEMBL8138162

SCHEMBL8138162

O=Cc1cncn1Cc1ccc(-c2cccc(F)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 12/20 0.55
CYP11B2 P19099 11/20 0.55
CYP17A1 P05093 1/20 0.50
CYP3A4 P08684 1/20 0.50
TAAR1 Q96RJ0 2/20 0.46
IDO1 P14902 1/20 0.43
GRM2 Q14416 1/20 0.42
HPGDS O60760 1/20 0.40
FNTA P49354 2/20 0.40
PGGT1B P53609 2/20 0.40
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7983220 0.87 CYP11B1 (0.62) CYP11B1CYP11B2IDO1FNTAPGGT1B
SCHEMBL5935193 0.85 CYP11B1 (0.63) CYP11B1CYP11B2CYP17A1IDO1HPGDS
SCHEMBL765399 0.82 CYP11B1 (0.67) CYP11B1CYP11B2IDO1
SCHEMBL7973153 0.81 CYP11B1 (0.58) CYP11B1CYP11B2CYP3A4IDO1GRM2
SCHEMBL8133106 0.80 CYP11B1 (0.63) CYP11B1CYP11B2IDO1FNTAPGGT1B
SCHEMBL14476244 0.78 CYP11B1 (0.58) CYP11B1CYP11B2IDO1FNTAPGGT1B
SCHEMBL1757759 0.76 CYP11B1 (0.66) CYP11B1CYP11B2IDO1HPGDS
SCHEMBL8135755 0.76 CYP11B1 (0.65) CYP11B1CYP11B2IDO1HPGDS
SCHEMBL8131698 0.75 CYP11B1 (0.58) CYP11B1CYP11B2IDO1GRM2
SCHEMBL7958104 0.75 CYP11B1 (0.58) CYP11B1CYP11B2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054882-A1 CONDENSED HETEROCYCLIC SYSTEM DERIVATIVES, PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Aventis Pharma S.A. (FR) 2000-11-29 EP disclosed
WO-1999041248-A1 CONDENSED HETEROCYCLIC SYSTEM DERIVATIVES, PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AVENTIS PHARMA S.A. (FR) 1999-08-19 WO disclosed