SCHEMBL8140480

SCHEMBL8140480

Cc1nc2c(=O)n(C)c(=O)n(Cc3ccco3)c2n1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.58
BLM P54132 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
MEN1 O00255 1/20 0.58
CYP1A1 P04798 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
NFKB1 P19838 1/20 0.58
MAPK1 P28482 1/20 0.58
CYP2C19 P33261 1/20 0.58
PMP22 Q01453 1/20 0.58
KMT2A Q03164 1/20 0.58
HIF1A Q16665 1/20 0.58
ADORA2A P29274 7/20 0.55
ADORA2B P29275 7/20 0.55
ALDH1A1 P00352 6/20 0.46
TSHR P16473 5/20 0.46
POLB P06746 4/20 0.44
MAPT P10636 4/20 0.44
NPSR1 Q6W5P4 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Furafylline SCHEMBL191214 0.73 MEN1 (1.00) LMNABLMSMN1; SMN2MEN1CYP1A1
SCHEMBL1457311 0.69 HTT (0.62) LMNABLMSMN1; SMN2MEN1CYP1A1
SCHEMBL23635735 0.69 ADORA2A (0.50) LMNABLMSMN1; SMN2MEN1CYP1A1
SCHEMBL2592397 0.69 TSHR (0.66) LMNABLMSMN1; SMN2MEN1CYP1A1
SCHEMBL15837498 0.68 TSHR (0.74) LMNABLMSMN1; SMN2MEN1CYP1A2
SCHEMBL9392263 0.68 MAPK1 (0.58) LMNABLMSMN1; SMN2MEN1CYP1A1
SCHEMBL15749615 0.66 ADORA2A (0.58) LMNABLMSMN1; SMN2MEN1CYP1A1
SCHEMBL15749716 0.66 HTT (0.60) LMNABLMSMN1; SMN2MEN1CYP1A1
SCHEMBL11279599 0.65 LMNA (0.57) LMNASMN1; SMN2MEN1MAPK1KMT2A
SCHEMBL9392090 0.64 TSHR (0.50) LMNABLMSMN1; SMN2MEN1CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6075029-A Xanthine modulators of metabolism of cellular P-450 CELL THERAPEUTICS, INC. (US) 2000-06-13 US disclosed