SCHEMBL8140679

SCHEMBL8140679

CSc1cc(N)nc(SCc2cccc3ccccc23)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
POLB P06746 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALPL P05186 1/20 0.43
MCL1 Q07820 1/20 0.42
HTT P42858 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
HSP90AA1 P07900 1/20 0.39
ABCB1 P08183 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8133994 0.85 RAB9A (0.39) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL8134849 0.85 CYP1A2 (0.55) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL8180602 0.84 RAB9A (0.43) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL6639259 0.81 NPC1 (0.48) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL6637576 0.81 NPC1 (0.48) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL8125033 0.81 ALDH1A1 (0.46) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL8138707 0.79 RAB9A (0.73) RAB9ANPC1SMN1; SMN2MEN1KMT2A
SCHEMBL8140098 0.77 RAB9A (0.54) RAB9ANPC1SMN1; SMN2LMNACYP1A2
SCHEMBL8136755 0.76 RAB9A (0.49) RAB9ANPC1SMN1; SMN2ALDH1A1MEN1
SCHEMBL8140696 0.75 CNR2 (0.41) RAB9ANPC1ALDH1A1HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124306-A Thioalkyl alpha substituted pyrimidine compounds PHARMACIA & UPJOHN COMPANY (US) 2000-09-26 US disclosed
EP-1034167-A1 ALPHA-ALKYLTHIO SUBSTITUTED PYRIMIDINE ETHERS AND THIOETHERS AS VIRAL REVERSE TRANSCRIPTASE INHIBITORS PHARMACIA & UPJOHN COMPANY (US) 2000-09-13 EP disclosed
WO-1999019304-A9 ALPHA-ALKYLTHIO SUBSTITUTED PYRIMIDINE ETHERS AND THIOETHERS AS VIRAL REVERSE TRANSCRIPTASE INHIBITORS UPJOHN CO (US) 1999-07-08 WO disclosed
WO-1999019304-A2 ALPHA-ALKYLTHIO SUBSTITUTED PYRIMIDINE ETHERS AND THIOETHERS AS VIRAL REVERSE TRANSCRIPTASE INHIBITORS PHARMACIA & UPJOHN COMPANY (US) 1999-04-22 WO disclosed