SCHEMBL8140689

SCHEMBL8140689

Cc1cc(I)cnc1Cl.Cc1cc(N)cnc1Cl

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
UHRF1 Q96T88 1/20 0.35
KDM4E B2RXH2 2/20 0.35
POLB P06746 1/20 0.33
IDO1 P14902 1/20 0.33
NOS3 P29474 2/20 0.32
NOS1 P29475 2/20 0.32
NOS2 P35228 2/20 0.32
CYP3A4 P08684 1/20 0.31
CHRNB2 P17787 5/20 0.31
CHRNA4 P43681 5/20 0.31
CHRNB4 P30926 4/20 0.31
CHRNA3 P32297 4/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4828775 0.88
SCHEMBL30135192 0.88
SCHEMBL1156177 0.88
SCHEMBL8125250 0.78 IDO1 (0.33) UHRF1IDO1NOS3NOS1NOS2
SCHEMBL8127902 0.77 ALDH1A1 (0.34) IDO1CYP3A4ALDH1A1
SCHEMBL7409028 0.71 ALDH1A1 (0.45) POLBIDO1CYP3A4ALDH1A1
SCHEMBL761151 0.71
SCHEMBL29437704 0.71
SCHEMBL3183893 0.71
SCHEMBL1722101 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970083-A1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-01-12 EP disclosed
WO-1998037082-A1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1998-08-27 WO disclosed