SCHEMBL8144398

SCHEMBL8144398

c1ccc2c(c1)CCCCN2.c1ccc2c(c1)CNCCN2

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD44 P16070 2/20 0.46
PNMT P11086 1/20 0.46
MAOB P27338 1/20 0.46
HTR2C P28335 6/20 0.41
HTR2B P41595 1/20 0.41
TSHR P16473 1/20 0.40
MAPT P10636 3/20 0.40
ALOX15 P16050 2/20 0.39
HSD17B10 Q99714 2/20 0.39
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
1,2,3,4-Tetrahydroisoquinoline SCHEMBL985673 0.88 PNMT (0.63) CD44PNMTMAOBHTR2CHTR2B
SCHEMBL28345077 0.87 TSHR (0.48) HTR2CTSHRMAPTALOX15HSD17B10
SCHEMBL28370547 0.87 TSHR (0.52) CD44PNMTMAOBHTR2CTSHR
SCHEMBL29373532 0.87 TSHR (0.52) CD44PNMTMAOBHTR2CTSHR
SCHEMBL24119 0.87 TSHR (0.52) CD44PNMTMAOBHTR2CTSHR
SCHEMBL379799 0.87 CD44 (0.52) CD44PNMTMAOBHTR2CALOX15
SCHEMBL6887634 0.87 CD44 (0.52) CD44PNMTMAOBHTR2CALOX15
SCHEMBL18320611 0.85 PNMT (0.47) CD44PNMTMAOBHTR2CALOX15
Hydrochloric Acid SCHEMBL7002945 0.85 CD44 (0.50) CD44PNMTMAOBHTR2CALOX15
SCHEMBL4504383 0.85 TSHR (0.50) HTR2CTSHRMAPTALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019383-A2 PROCESS FOR THE AMINOCARBONYLATION OF BENZAZEPINES AND BENZODIAZEPINES SMITHKLINE BEECHAM PLC (GB) 2000-07-19 EP disclosed
WO-1997024336-A2 PROCESS FOR THE AMINOCARBONYLATION OF BENZAZEPINES AND BENZODIAZEPINES SMITHKLINE BEECHAM PLC (GB) 1997-07-10 WO disclosed