SCHEMBL8147306

SCHEMBL8147306

COc1c(Cl)cc(C(F)(F)F)c(C(=O)O)c1N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 1/20 0.45
TPMT P51580 1/20 0.42
MAPT P10636 4/20 0.40
LMNA P02545 3/20 0.39
GAA P10253 2/20 0.39
MEN1 O00255 2/20 0.37
HTT P42858 2/20 0.37
KMT2A Q03164 2/20 0.37
TMPRSS4 Q9NRS4 1/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL609987 0.81 ALDH1A1 (0.53) ALDH1A1KDM4EHSD17B10TPMTLMNA
SCHEMBL14960283 0.80 ALDH1A1 (0.51) ALDH1A1KDM4EHSD17B10TPMTLMNA
SCHEMBL8156118 0.78 TTR (0.40) ALDH1A1KDM4EHSD17B10GABRPGABRD
SCHEMBL28883701 0.74 ALDH1A1 (0.58) ALDH1A1KDM4EHSD17B10TPMTLMNA
SCHEMBL1458336 0.74 TPMT (0.61) ALDH1A1KDM4EHSD17B10TPMTMAPT
SCHEMBL1323406 0.71 ALDH1A1 (0.68) ALDH1A1KDM4EHSD17B10TPMTLMNA
SCHEMBL9769182 0.71 MAPT (0.39) ALDH1A1KDM4EHSD17B10MAPTGAA
SCHEMBL22061113 0.71 ALDH1A1 (0.49) ALDH1A1KDM4EHSD17B10TPMTMAPT
SCHEMBL1633542 0.71 CA12 (0.44) ALDH1A1KDM4ETPMTMAPTLMNA
SCHEMBL613131 0.70 KDM4E (0.47) ALDH1A1KDM4EHSD17B10TPMTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686145-B1 NEW COMPOUNDS UNIV MARYLAND (US) 2000-01-26 EP disclosed
US-5883129-A Hydroxylated anthranilic acid derivatives ASTRA AKTIEBOLAG (SE) 1999-03-16 US disclosed
US-5523475-A New compounds AKTIEBOLAGET ASTRA (SE) 1996-06-04 US disclosed
EP-0686145-A1 NEW COMPOUNDS AKTIEBOLAGET ASTRA (SE) 1995-12-13 EP disclosed
WO-1994019316-A1 NEW COMPOUNDS AKTIEBOLAGET ASTRA (SE) 1994-09-01 WO disclosed