SCHEMBL8148012

SCHEMBL8148012

CN1CCc2ccc(NC(=O)Nc3cccc(Br)c3)cc2C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.56
GAA P10253 1/20 0.56
PRMT5 O14744 1/20 0.54
WDR77 Q9BQA1 1/20 0.54
NPC1 O15118 6/20 0.51
RAB9A P51151 6/20 0.51
ROCK2 O75116 4/20 0.50
L3MBTL3 Q96JM7 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
CASP3 P42574 2/20 0.48
SENP7 Q9BQF6 2/20 0.48
CYP3A4 P08684 2/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
PKM P14618 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
THPO P40225 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8130701 0.87 NPC1 (0.65) NPC1RAB9AROCK2MEN1KMT2A
SCHEMBL8128776 0.85 MAPT (0.60) GAAPRMT5WDR77NPC1RAB9A
SCHEMBL8126912 0.85 RAB9A (0.68) GAAPRMT5WDR77NPC1RAB9A
Hydrochloric Acid SCHEMBL8128910 0.85 NPC1 (0.53) NPC1RAB9AROCK2MEN1KMT2A
SCHEMBL8133044 0.85 NPC1 (0.70) KDM4EPRMT5WDR77NPC1RAB9A
SCHEMBL8120020 0.85 DDX3X (0.57) NPC1RAB9AROCK2MEN1KMT2A
SCHEMBL8130811 0.83 KDM4E (0.52) KDM4EGAAPRMT5WDR77MEN1
SCHEMBL8155988 0.83 RAF1 (0.49) NPC1RAB9AROCK2MEN1KMT2A
SCHEMBL8132666 0.83 NPC1 (0.72) KDM4ENPC1RAB9AMEN1KMT2A
SCHEMBL8131782 0.83 MAPT (0.59) KDM4ENPC1RAB9AROCK2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1005459-A1 SUBSTITUTED ISOQUINOLINES AS ANTICONVULSIVANTS SMITHKLINE BEECHAM PLC (GB) 2000-06-07 EP disclosed
WO-1999014197-A1 SUBSTITUTED ISOQUINOLINES AS ANTICONVULSIVANTS SMITHKLINE BEECHAM PLC (GB) 1999-03-25 WO disclosed