SCHEMBL8148995

SCHEMBL8148995

N#Cc1cccc(N)c1CN1CCCCC1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.47
HRH3 Q9Y5N1 1/20 0.41
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
TSHR P16473 1/20 0.38
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CYP2D6 P10635 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
ACHE P22303 1/20 0.36
ACACB O00763 1/20 0.36
KLKB1 P03952 1/20 0.35
GRM2 Q14416 1/20 0.35
CYP3A4 P08684 1/20 0.34
PER2 O15055 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8144666 0.95 MAPK1 (0.41) L3MBTL1HRH3MAPK1KMT2ATSHR
SCHEMBL248961 0.79 KDM4E (0.48) HRH3TSHRCYP1A2CYP2C9CYP2C19
SCHEMBL20576177 0.70 L3MBTL1 (0.64) L3MBTL1HRH3ACHEACACBGRM2
SCHEMBL249557 0.70 CYP2A13 (0.50) HRH3KMT2ACYP2C9KDM4EALDH1A1
Hydrochloric Acid SCHEMBL12494160 0.69 L3MBTL1 (0.55) L3MBTL1HRH3MAPK1KMT2AACHE
SCHEMBL6737403 0.68 CYP3A4 (0.43) KMT2ATSHRCYP1A2CYP2C9CYP2C19
SCHEMBL14537170 0.68 MAPK1 (0.56) L3MBTL1HRH3MAPK1KMT2ATSHR
SCHEMBL2222171 0.68 L3MBTL1 (0.65) L3MBTL1HRH3MAPK1KMT2AACHE
SCHEMBL2223756 0.67 L3MBTL1 (0.70) L3MBTL1HRH3MAPK1KMT2ACYP1A2
SCHEMBL20505562 0.67 ACACB (0.60) L3MBTL1HRH3CYP1A2CYP2C9ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853618-A4 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2000-03-15 EP disclosed
EP-0853618-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1998-07-22 EP disclosed