SCHEMBL8149641

SCHEMBL8149641

O=C1CCCCN1c1ccc(CO)cc1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
HPGD P15428 4/20 0.54
USP2 O75604 2/20 0.51
MAPT P10636 4/20 0.50
LMNA P02545 2/20 0.50
AKR1C3 P42330 2/20 0.50
ACACB O00763 1/20 0.49
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47
BLM P54132 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
RECQL P46063 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14473350 0.96 ALDH1A1 (0.62) ALDH1A1HPGDUSP2MAPTLMNA
SCHEMBL8330770 0.92 ALDH1A1 (0.50) ALDH1A1HPGDUSP2MAPTLMNA
SCHEMBL12676673 0.86 ALDH1A1 (0.54) ALDH1A1HPGDUSP2MAPTLMNA
SCHEMBL1907807 0.83 ALDH1A1 (0.58) ALDH1A1HPGDUSP2MAPTLMNA
SCHEMBL1696787 0.82 USP2 (0.55) ALDH1A1HPGDUSP2MAPTLMNA
SCHEMBL8154285 0.82 ALDH1A1 (0.53) ALDH1A1HPGDUSP2MAPTLMNA
SCHEMBL79080 0.82 ALDH1A1 (0.53) ALDH1A1HPGDUSP2MAPTLMNA
SCHEMBL21770514 0.82 ALDH1A1 (0.53) ALDH1A1HPGDUSP2MAPTLMNA
SCHEMBL2644969 0.81 ALDH1A1 (0.61) ALDH1A1HPGDUSP2MAPTLMNA
SCHEMBL6788342 0.81 ALDH1A1 (0.61) ALDH1A1HPGDUSP2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12016852-B2 Pyrrolidine glycosidase inhibitors ASCENEURON SA (CH) 2024-06-25 US disclosed
US-12016852-B2 Pyrrolidine glycosidase inhibitors ASCENEURON SA (CH) 2024-06-25 US disclosed
US-20210213005-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS ASCENEURON SA (CH) 2021-07-15 US disclosed
US-20210213005-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS ASCENEURON SA (CH) 2021-07-15 US disclosed
WO-2020039027-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS ASCENEURON S. A. (CH) 2020-02-27 WO disclosed
WO-2020039027-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS ASCENEURON S. A. (CH) 2020-02-27 WO disclosed
US-6077853-A Inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 2000-06-20 US disclosed
EP-0951285-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-10-27 EP disclosed
US-5939439-A Inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 1999-08-17 US disclosed
WO-1998029119-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1998-07-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12016852-B2 Pyrrolidine glycosidase inhibitors PREP, GAA, DNPEP ALDH1A1 1182/4885HPGD 1673/4885USP2 2385/4885
US-20210213005-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS PREP, GAA, DNPEP ALDH1A1 1170/4885HPGD 1675/4885USP2 2309/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.