SCHEMBL8150384

SCHEMBL8150384

CCOC(=O)c1ccc(-c2ccc(N3CCCC3=O)cc2CO)cc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.55
HSD17B10 Q99714 1/20 0.55
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
HPGD P15428 3/20 0.48
TSHR P16473 2/20 0.48
LMNA P02545 2/20 0.48
MAPT P10636 4/20 0.46
ALDH1A1 P00352 4/20 0.45
USP2 O75604 1/20 0.43
GLA P06280 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HTT P42858 1/20 0.43
CACNA1B Q00975 1/20 0.43
APBA1 Q02410 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8140892 0.91 PKM (0.52) PKMHSD17B10NPC1RAB9ARXFP1
SCHEMBL4196712 0.84 PKM (0.67) PKMHSD17B10NPC1RAB9ARXFP1
SCHEMBL14686859 0.80 PKM (0.63) PKMHSD17B10NPC1RAB9ARXFP1
SCHEMBL5515479 0.79 MAPT (0.51) NPC1RAB9AHPGDTSHRLMNA
SCHEMBL25236156 0.79 PKM (0.62) PKMHSD17B10NPC1RAB9ARXFP1
SCHEMBL8134923 0.78 HPGD (0.50) NPC1RAB9ARXFP1HPGDTSHR
SCHEMBL7431121 0.76 HTT (0.57) PKMHSD17B10NPC1RAB9ARXFP1
SCHEMBL8143968 0.75 ALDH1A1 (0.47) NPC1RAB9ARXFP1HPGDTSHR
SCHEMBL8144130 0.75 ATM (0.52) NPC1RAB9ARXFP1HPGDTSHR
SCHEMBL8135805 0.75 ALDH1A1 (0.65) HPGDTSHRLMNAALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100272-A Tetracyclic spiro compounds as 5HT1B receptor antagonists SMITHKLINE BEECHAM P.L.C. (GB) 2000-08-08 US disclosed
EP-0888358-A1 PIPERIDINE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 1999-01-07 EP disclosed
WO-1997034901-A1 PIPERIDINE DERIVATIVES SMITHKLINE BEECHAM P.L.C. (GB) 1997-09-25 WO disclosed