SCHEMBL8151691

SCHEMBL8151691

C=C[C@]1(O)CC[C@H]2[C@@H]3CCc4cc(OCCN(C)C)ccc4[C@H]3CC[C@@]21C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.53
ESR2 Q92731 2/20 0.53
NR3C1 P04150 4/20 0.52
LMNA P02545 3/20 0.52
PGR P06401 2/20 0.52
CYP2C19 P33261 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
HIF1A Q16665 1/20 0.52
CNR1 P21554 1/20 0.52
SLC6A2 P23975 1/20 0.52
SLC6A4 P31645 1/20 0.52
SLC6A3 Q01959 1/20 0.52
STS P08842 10/20 0.49
MAPT P10636 2/20 0.49
GAA P10253 1/20 0.49
MAPK1 P28482 1/20 0.49
NR3C2 P08235 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP2C9 P11712 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8151660 0.96 ESR1 (0.52) ESR1ESR2NR3C1LMNAPGR
SCHEMBL8145946 0.88 STS (0.64) ESR1NR3C1LMNAPGRCYP2C19
SCHEMBL8151948 0.86 STS (0.67) ESR1NR3C1LMNAPGRCYP2C19
SCHEMBL8145976 0.86 ESR1 (0.55) ESR1ESR2NR3C1LMNAPGR
SCHEMBL8145253 0.86 ESR1 (0.55) ESR1ESR2NR3C1LMNAPGR
SCHEMBL8158827 0.85 ESR1 (0.73) ESR1ESR2NR3C1LMNAPGR
SCHEMBL8159727 0.83 STS (0.62) ESR1NR3C1LMNAPGRCYP2C19
SCHEMBL1656677 0.82 ESR1 (0.63) ESR1ESR2NR3C1LMNAPGR
SCHEMBL4645148 0.82 ESR1 (0.63) ESR1ESR2NR3C1LMNAPGR
SCHEMBL8151131 0.82 STS (0.66) ESR1NR3C1LMNAPGRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676202-B1 Use of aromatic steroids substituted in 3-position by a disubstituted aminoalkoxy chain for the manufacture of a medicament for the control of fertility, in particular male fertility HOECHST MARION ROUSSEL INC (FR) 2000-06-07 EP claimed