SCHEMBL8152227

SCHEMBL8152227

COc1ccccc1N1CCC1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.52
MGLL Q99685 1/20 0.51
DRD2 P14416 2/20 0.50
DRD3 P35462 2/20 0.50
MAPT P10636 2/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP1A2 P05177 1/20 0.49
HTR1A P08908 1/20 0.49
CYP2C9 P11712 1/20 0.49
HTR7 P34969 1/20 0.49
ALDH1A1 P00352 2/20 0.49
POLB P06746 1/20 0.49
HTR3E A5X5Y0 1/20 0.49
HTR3B O95264 1/20 0.49
ADRB1 P08588 1/20 0.49
HTR3A P46098 1/20 0.49
HTR6 P50406 1/20 0.49
HTR3D Q70Z44 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1829260 0.90 MAPT (0.58) ATMMGLLDRD2DRD3MAPT
SCHEMBL1624631 0.88 MAPT (0.54) ATMMGLLDRD2DRD3MAPT
SCHEMBL25575695 0.80 CRBN (0.65) ATMMGLLDRD2DRD3MAPT
SCHEMBL30160700 0.80 CRBN (0.65) ATMMGLLDRD2DRD3MAPT
SCHEMBL12989510 0.80 ATM (0.48) ATMMGLLDRD2DRD3MAPT
SCHEMBL11819234 0.79 SMN1; SMN2 (0.50) DRD2DRD3MAPTMEN1KMT2A
SCHEMBL8276483 0.79 DRD2 (0.58) ATMMGLLDRD2DRD3MAPT
SCHEMBL7958379 0.79 GSK3A (0.56) DRD2DRD3MAPTCYP2C19ALDH1A1
SCHEMBL23356608 0.78 GAA (0.58) DRD2DRD3HTR7ALDH1A1POLB
Hydrochloric Acid SCHEMBL10705356 0.78 ATM (0.59) ATMMGLLDRD2DRD3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944594-A4 INHIBITORS OF THE ENZYMATIC ACTIVITY OF PSA LILLY CO ELI (US) 2000-05-03 EP disclosed
EP-0944594-A1 INHIBITORS OF THE ENZYMATIC ACTIVITY OF PSA ELI LILLY AND COMPANY (US) 1999-09-29 EP disclosed
WO-1998025895-A1 INHIBITORS OF THE ENZYMATIC ACTIVITY OF PSA ELI LILLY AND COMPANY (US) 1998-06-18 WO disclosed