SCHEMBL30160700

SCHEMBL30160700

COc1ccccc1N1CCC(=O)NC1=O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 7/20 0.65
DDB1 Q16531 6/20 0.65
ALDH1A1 P00352 1/20 0.51
POLB P06746 1/20 0.51
ATM Q13315 1/20 0.51
GSK3A P49840 1/20 0.48
GSK3B P49841 1/20 0.48
DRD2 P14416 2/20 0.47
DRD3 P35462 2/20 0.47
CYP2C19 P33261 2/20 0.47
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
ADRB1 P08588 1/20 0.47
HTR3A P46098 1/20 0.47
HTR6 P50406 1/20 0.47
HTR3D Q70Z44 1/20 0.47
HTR3C Q8WXA8 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
MAPT P10636 2/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25575695 1.00 CRBN (0.65) CRBNDDB1ALDH1A1POLBATM
Trifluoroacetic Acid SCHEMBL30874158 0.88 DDB1 (0.52) CRBNDDB1ALDH1A1POLBATM
SCHEMBL25575719 0.84 CRBN (0.60) CRBNDDB1ALDH1A1DRD2DRD3
SCHEMBL24777726 0.82 HTR3E (0.52) CRBNDDB1ALDH1A1POLBHTR3E
SCHEMBL25653902 0.82 CRBN (0.48) CRBNDDB1ATM
SCHEMBL29547244 0.82 GSK3B (0.53) CRBNDDB1ALDH1A1POLBATM
SCHEMBL25905651 0.81 CRBN (0.56) CRBNDDB1
SCHEMBL23065973 0.81 DDB1 (0.52) CRBNDDB1ALDH1A1MAPTLMNA
SCHEMBL8152227 0.80 ATM (0.52) ALDH1A1POLBATMDRD2DRD3
SCHEMBL24155758 0.80 NTRK1 (0.52) CRBNDDB1ALDH1A1HTR6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240261416-A1 SYNTHESIS OF NOVEL CEREBLON E3 LIGASE LIGANDS, COMPOUNDS FORMED THEREBY, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2024-08-08 US disclosed
WO-2023274390-A1 BRUTON'S TYROSINE KINASE AND MUTANT DEGRADER, COMPOSITION AND APPLICATION THEREOF 杭州和正医药有限公司 2023-01-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240261416-A1 SYNTHESIS OF NOVEL CEREBLON E3 LIGASE LIGANDS, COMPOUNDS FORMED THEREBY, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM CRBN, CUL1, CUL5 CRBN 1/4885DDB1 188/4885ALDH1A1 2015/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.