SCHEMBL8152855

SCHEMBL8152855

C=C1/C(=C\C=C2/CCC[C@]3(C)[C@@H]([C@H](C)CCC(=O)C(C)C)CC[C@@H]23)C[C@@H](O)CC1O

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VDR P11473 14/20 0.76
ADORA3 P0DMS8 2/20 0.76
SLC6A2 P23975 2/20 0.76
AGTR1 P30556 2/20 0.76
CYP24A1 Q07973 3/20 0.73
MAPT P10636 2/20 0.73
NR1I2 O75469 1/20 0.73
ABCB11 O95342 1/20 0.73
GC P02774 1/20 0.73
PGR P06401 1/20 0.73
RXRA P19793 1/20 0.73
CHRM3 P20309 1/20 0.73
CNR1 P21554 1/20 0.73
HTR2C P28335 1/20 0.73
MAPK1 P28482 1/20 0.73
SLC6A4 P31645 1/20 0.73
ADRA1A P35348 1/20 0.73
PTGS2 P35354 1/20 0.73
OPRD1 P41143 1/20 0.73
OPRK1 P41145 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7080225 1.00 VDR (0.76) VDRADORA3SLC6A2AGTR1CYP24A1
SCHEMBL30013587 1.00 VDR (0.76) VDRADORA3SLC6A2AGTR1CYP24A1
SCHEMBL26982954 1.00 VDR (0.76) VDRADORA3SLC6A2AGTR1CYP24A1
SCHEMBL7080227 1.00 VDR (0.76) VDRADORA3SLC6A2AGTR1CYP24A1
SCHEMBL3679281 0.92 VDR (0.83) VDRADORA3SLC6A2AGTR1CYP24A1
SCHEMBL29452954 0.90 VDR (0.75) VDRADORA3SLC6A2AGTR1CYP24A1
SCHEMBL19988215 0.90 VDR (0.79) VDRADORA3SLC6A2AGTR1CYP24A1
SCHEMBL8046820 0.90 VDR (0.79) VDRADORA3SLC6A2AGTR1CYP24A1
SCHEMBL7139484 0.90 VDR (0.79) VDRADORA3SLC6A2AGTR1CYP24A1
SCHEMBL19988232 0.90 VDR (0.79) VDRADORA3SLC6A2AGTR1CYP24A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0969849-A1 STABLE SOLID PREPARATION CONTAINING VITAMIN D3 AND TRICALCIUM PHOSPHATE MERCK PATENT GmbH (DE) 2000-01-12 EP disclosed
WO-1998040085-A1 STABLE SOLID PREPARATION CONTAINING VITAMIN D3 AND TRICALCIUM PHOSPHATE MERCK PATENT GMBH (DE) 1998-09-17 WO disclosed
US-4292249-A VITAMIN D3 INTERMEDIATES TEIJIN LIMITED (JP) 1981-09-29 US disclosed
EP-0015122-A1 New 25-hydroxy-24-oxocholestane derivatives and preparation thereof TEIJIN LIMITED (JP) 1980-09-03 EP disclosed